TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 33.8nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 557nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 580nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 1.08E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 1.57E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 1.97E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 2.65E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.13E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.40E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.94E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 4.70E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 5.03E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 7.40E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 9.83E+3nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 1.70E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 2.20E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 2.49E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 2.61E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 2.92E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 2.99E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.05E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.15E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.33E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.61E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.61E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 3.79E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 4.51E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 6(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 4.71E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair
TargetHistone deacetylase 3(Homo sapiens (Human))
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
The Royal Institution For The Advancement Of Learning/Mcgill University
US Patent
Affinity DataIC50: 4.73E+4nMpH: 8.1 T: 2°CAssay Description:Boc-Lys(Ac)-7-amino-4-methylcoumarin (Boc-Lys(Ac)-AMC) was used as substrate for the HDAC assays. Substrate solution was prepared as follow: Boc(Lys-...More data for this Ligand-Target Pair