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Found 32 with Last Name = 'kamiyasu' and Initial = 'k'
TargetSerine protease 1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50:  4.13nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Boc-Phe-Ser-Arg-AMC) for trypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50:  11.2nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Boc-Phe-Ser-Arg-AMC) for trypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50:  50.6nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Boc-Phe-Ser-Arg-AMC) for trypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50:  55nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Boc-Phe-Ser-Arg-AMC) for trypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50:  97nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Pro-Phe-Arg-pNA) for plasma kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50:  190nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Pro-Phe-Arg-pNA) for plasma kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50:  873nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50:  1.48E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Pro-Phe-Arg-pNA) for plasma kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50:  1.83E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50:  2.32E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Pro-Phe-Arg-pNA) for plasma kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50:  2.62E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50:  3.66E+3nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Phe-Pip-Arg-pNA) thrombin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Rattus norvegicus)
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50:  1.25E+4nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Lys-pNA) for plasmin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50:  1.57E+4nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Arg-pNA) for pancreatic kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50:  3.16E+4nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Phe-Pip-Arg-pNA) thrombin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50:  3.41E+4nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Arg-pNA) for pancreatic kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50:  3.50E+4nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Phe-Pip-Arg-pNA) thrombin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Met-pNA) for cathepsin G in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Suc-Ala-Ala-Pro-Phe-pNA) for chymotrypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Met-pNA) for cathepsin G in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Val-pNA) for sputum elastase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Suc-Ala-Ala-Pro-Phe-pNA) for chymotrypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Met-pNA) for cathepsin G in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Val-pNA) for sputum elastase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031708(4-[(E)-2-(Allyl-ethoxycarbonylmethyl-carbamoyl)-pr...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Suc-Ala-Ala-Pro-Phe-pNA) for chymotrypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin G(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Met-pNA) for cathepsin G in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChymotrypsinogen A(Bos taurus (bovine))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (Suc-Ala-Ala-Pro-Phe-pNA) for chymotrypsin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031706(4-Guanidino-benzoic acid 4-dimethylcarbamoylmethox...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Val-pNA) for sputum elastase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031707(4-[(E)-2-(Allyl-carboxymethyl-carbamoyl)-propenyl]...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Arg-pNA) for pancreatic kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (MeO-Suc-Ala-Ala-Pro-Val-pNA) for sputum elastase in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50: >1.00E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Val-Leu-Arg-pNA) for pancreatic kallikrein in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Minase Research Institute

Curated by ChEMBL
LigandPNGBDBM50031709(4-Guanidino-benzoic acid 4-carboxymethyl-phenyl es...)
Affinity DataIC50:  1.08E+5nMAssay Description:Concentration required to inhibit enzymatic cleavage of the chromogenic substrate (H-D-Phe-Pip-Arg-pNA) thrombin in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed