Affinity DataKi: 0.211nMAssay Description:Inhibition of BRD4 in human HL60 cells assessed as reduction in C-myc production after 24 hrs by ELISAMore data for this Ligand-Target Pair
Affinity DataKi: 0.221nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKi: 0.265nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKi: 0.313nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.336nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.356nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.362nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.455nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.458nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.479nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.522nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.545nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.564nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.578nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.585nMAssay Description:Inhibition of recombinant human N-terminal His-tagged BRD4 bromodomain 1 (49 to 170 residues) expressed in Escherichia coli using biotinylated peptid...More data for this Ligand-Target Pair
Affinity DataKi: 0.610nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 0.670nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 0.726nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.75nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.75nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.781nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.790nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.813nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.826nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.833nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.940nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.950nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.953nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKi: 0.970nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 0.990nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 2nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair