Compile Data Set for Download or QSAR
maximum 50k data
Found 202 with Last Name = 'kanda' and Initial = 't'
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataKi:  0.211nMAssay Description:Inhibition of BRD4 in human HL60 cells assessed as reduction in C-myc production after 24 hrs by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataKi:  0.221nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataKi:  0.265nMAssay Description:Agonist activity at human recombinant KOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataKi:  0.313nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataKi:  0.336nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataKi:  0.356nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataKi:  0.362nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254124(CHEMBL4103044)
Affinity DataKi:  0.455nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataKi:  0.458nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataKi:  0.479nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataKi:  0.522nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179992(US9676720, Example 2)
Affinity DataKi:  0.530nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254133(CHEMBL4076632)
Affinity DataKi:  0.545nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataKi:  0.564nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254132(CHEMBL4083940)
Affinity DataKi:  0.578nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254130(CHEMBL4061334)
Affinity DataKi:  0.585nMAssay Description:Inhibition of recombinant human N-terminal His-tagged BRD4 bromodomain 1 (49 to 170 residues) expressed in Escherichia coli using biotinylated peptid...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179995(US9676720, Example 7)
Affinity DataKi:  0.610nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290167(1,3-Diethyl-8-[(E)-2-(4-methoxy-2,3-dimethyl-pheny...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290165(8-[(E)-2-(2,4-Dimethoxy-3-methyl-phenyl)-vinyl]-1,...)
Affinity DataKi:  0.670nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254123(CHEMBL4068691)
Affinity DataKi:  0.726nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179994(US9676720, Example 6)
Affinity DataKi:  0.75nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180045(US9676720, Comparative example 16)
Affinity DataKi:  0.75nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetKappa-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataKi:  0.781nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179998(US9676720, Example 11)
Affinity DataKi:  0.790nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179993(US9676720, Example 4)
Affinity DataKi:  0.800nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179996(US9676720, Example 9)
Affinity DataKi:  0.800nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254131(CHEMBL4094845)
Affinity DataKi:  0.813nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataKi:  0.826nMAssay Description:Displacement of [3H]DAMGO from human recombinant MOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254120(CHEMBL4076681)
Affinity DataKi:  0.833nMAssay Description:Displacement of [3H]DPDPE from human recombinant DOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180000(US9676720, Example 14)
Affinity DataKi:  0.900nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179999(US9676720, Example 12)
Affinity DataKi:  0.940nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180002(US9676720, Example 16)
Affinity DataKi:  0.950nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMu-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataKi:  0.953nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM179997(US9676720, Example 10)
Affinity DataKi:  0.970nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180003(US9676720, Example 18)
Affinity DataKi:  0.990nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006710(8-[(E)-2-(3,4-Dimethoxy-phenyl)-vinyl]-7-methyl-1,...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180020(US9676720, Comparative example 8)
Affinity DataKi:  1.10nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180024(US9676720, Comparative example 11)
Affinity DataKi:  1.20nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254121(CHEMBL4067629)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]U-69,593 from human recombinant KOR expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180019(US9676720, Comparative example 7)
Affinity DataKi:  1.40nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180004(US9676720, Example 19)
Affinity DataKi:  1.40nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180021(US9676720, Comparative example 9)
Affinity DataKi:  1.5nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180005(US9676720, Comparative example 1)
Affinity DataKi:  1.5nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetDelta-type opioid receptor(Homo sapiens (Human))
Nippon Chemiphar

Curated by ChEMBL
LigandPNGBDBM50254122(CHEMBL4098662)
Affinity DataKi:  1.5nMAssay Description:Agonist activity at human recombinant DOR expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290165(8-[(E)-2-(2,4-Dimethoxy-3-methyl-phenyl)-vinyl]-1,...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]-CHA from Adenosine A1 receptor of rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50006714(7-Methyl-1,3-dipropyl-8-[(E)-2-(3,4,5-trimethoxy-p...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180022(US9676720, Comparative example 10)
Affinity DataKi:  1.70nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180025(US9676720, Comparative example 12)
Affinity DataKi:  2nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50290167(1,3-Diethyl-8-[(E)-2-(4-methoxy-2,3-dimethyl-pheny...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-CGS- 21680 from Adenosine A2a receptor of rat forebrain membranes (shielded from light)More data for this Ligand-Target Pair
In DepthDetails Article
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Ube Industries

US Patent
LigandPNGBDBM180018(US9676720, Comparative example 6)
Affinity DataKi:  2.20nMpH: 6.0Assay Description:Measurement of EP2 receptor binding action was performed in accordance with the method of Abramovitz et al. (Biochimica et Biophysica Acta, 1483, 285...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 202 total ) | Next | Last >>
Jump to: