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Found 129 with Last Name = 'kaneko' and Initial = 'y'
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427221(5-Aminonicotinic Acid | CHEMBL1491941)
Affinity DataKi:  3.80E+3nMAssay Description:Binding affinity to human recombinant DDOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRCG38204, isoform CRA_d(Rattus norvegicus)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427221(5-Aminonicotinic Acid | CHEMBL1491941)
Affinity DataKi:  5.89E+3nMAssay Description:Inhibition of rat recombinant DDO using D-AspMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Mus musculus)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427221(5-Aminonicotinic Acid | CHEMBL1491941)
Affinity DataKi:  8.69E+3nMAssay Description:Inhibition of mouse recombinant DDO using D-AspMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121995(CHEMBL3617316)
Affinity DataKi:  1.51E+4nMAssay Description:Binding affinity to human recombinant DDOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Mus musculus)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121995(CHEMBL3617316)
Affinity DataKi:  3.26E+4nMAssay Description:Inhibition of mouse recombinant DDO using D-AspMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRCG38204, isoform CRA_d(Rattus norvegicus)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121995(CHEMBL3617316)
Affinity DataKi:  6.59E+4nMAssay Description:Inhibition of rat recombinant DDO using D-AspMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  1.53E+5nMAssay Description:Binding affinity to human recombinant DDOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Mus musculus)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  1.22E+6nMAssay Description:Inhibition of mouse recombinant DDO using D-AspMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRCG38204, isoform CRA_d(Rattus norvegicus)
Kitasato University

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataKi:  1.56E+6nMAssay Description:Inhibition of rat recombinant DDO using D-AspMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50132151(CHEMBL101683 | N-(4-Chloro-phenyl)-2-[(pyridin-4-y...)
Affinity DataIC50:  20nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM9503(2-[(pyridin-4-ylmethyl)amino]-N-[3-(trifluoromethy...)
Affinity DataIC50:  23nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377602(CHEMBL256556)
Affinity DataIC50:  26nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM4851((4-chlorophenyl)-[4-(4-pyridylmethyl)phthalazin-1-...)
Affinity DataIC50:  37nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377603(CHEMBL402002)
Affinity DataIC50:  46nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377606(CHEMBL427725)
Affinity DataIC50:  200nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593237(CHEMBL5199411)
Affinity DataIC50:  500nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593236(CHEMBL5185636)
Affinity DataIC50:  850nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377604(CHEMBL256718)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Santen Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50377605(CHEMBL404393)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of KDR by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122008(CHEMBL3617314)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593235(CHEMBL5180151)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593234(CHEMBL5208116)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593233(CHEMBL5173170)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593232(CHEMBL5194442)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593230(CHEMBL5170507)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50427221(5-Aminonicotinic Acid | CHEMBL1491941)
Affinity DataIC50:  2.19E+4nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593231(CHEMBL5180122)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593231(CHEMBL5180122)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593229(CHEMBL5196345)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121995(CHEMBL3617316)
Affinity DataIC50:  8.71E+4nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121998(CHEMBL3322866)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121997(CHEMBL3322863)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121996(CHEMBL3617326)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122001(CHEMBL3617320)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121998(CHEMBL3322866)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121996(CHEMBL3617326)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121997(CHEMBL3322863)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122001(CHEMBL3617320)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593228(CHEMBL5174487)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM197302(Benzoic acid | SAMPL4, O1)
Affinity DataIC50:  1.34E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122006(CHEMBL3617317)
Affinity DataIC50:  3.47E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50226518(3-Aminobenzoesaeure | 3-aminobenzoic acid | CHEMBL...)
Affinity DataIC50:  3.92E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50121995(CHEMBL3617316)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM14673(Fragment 3 | Malonic Acid | propanedioic acid)
Affinity DataIC50:  8.79E+5nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122008(CHEMBL3617314)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122003(CHEMBL3617319)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122000(CHEBI:68572 | CHEMBL3322868)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122003(CHEMBL3617319)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Astex Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50593238(CHEMBL5174785)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of full length recombinant C-terminal FLAG-tagged human HDAC2 expressed in baculovirus-infected Sf9 cells measured for 2 hrs by fluorescen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD-aspartate oxidase(Homo sapiens (Human))
Kitasato University

Curated by ChEMBL
LigandPNGBDBM50122000(CHEBI:68572 | CHEMBL3322868)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of human recombinant DDO expressed in Escherichia coli BL21(DE3) using D-Asp and D-Ala assessed as 2-oxo acid production after 10 mins by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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