Compile Data Set for Download or QSAR
maximum 50k data
Found 16 with Last Name = 'karle' and Initial = 'jm'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50201426(dispiro[adamantane-2,2'-[1,3,5]trioxolane-4',1''-c...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of hERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50201425(2-({dispiro[adamantane-2,2'-[1,3,5]trioxolane-4',1...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of hERG by patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM22985(Aralen | CHEMBL76 | CHLOROQUINE PHOSPHATE | Chloro...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408762(DESETHYLCHLOROQUINE | Desethyl chloroquine)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408763(CHEMBL343728)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM23300(4-amino-7-chloroquinoline (ACQ)-based compound, 5 ...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408770(CHEMBL143042 | TCMDC-124246)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408771(CHEMBL344599)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408760(CHEMBL139984)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408766(CHEMBL342499)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408768(CHEMBL423184)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408764(CHEMBL143439)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408761(CHEMBL143522)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408769(CHEMBL142884)
Affinity DataIC50: >2.50E+6nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408765(CHEMBL143331)
Affinity DataIC50: >2.50E+6nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistidine-rich protein PFHRP-II(Plasmodium falciparum)
University Of Nebraska Medical Center

Curated by ChEMBL
LigandPNGBDBM50408767(CHEMBL143177)
Affinity DataIC50: >2.50E+6nMAssay Description:Inhibition of hematin polymerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed