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Found 20 with Last Name = 'kathiravan' and Initial = 'mk'
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50029257((3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)p...)
Affinity DataKi:  0.0200nMAssay Description:Binding affinity to adrenergic alpha1A receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50270453((R)-4-(3-(2-amino-4-(4-fluorophenyl)thiazol-5-yl)p...)
Affinity DataKi:  1.92nMAssay Description:Binding affinity to 5HT2A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50029257((3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)p...)
Affinity DataKi:  47nMAssay Description:Binding affinity to adrenergic alpha1B receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol 14-alpha demethylase(Rattus norvegicus)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213693((3S,5S,8R,9S,10S,13R,14R,17R)-5,13-dimethyl-17-((R...)
Affinity DataKi:  600nMAssay Description:Inhibition of rat liver LDMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-citrate synthase(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50066683((S)-2-((R)-8-(2,4-dichlorophenyl)-2-hydroxyoctyl)-...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human ATP citrate lyaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50029257((3-((4-(2-isopropoxyphenyl)piperazin-1-yl)methyl)p...)
Affinity DataKi:  2.88E+3nMAssay Description:Binding affinity to 5HT1B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Candida albicans (strain SC5314 / ATCC MYA-2876) (...)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055641(2,2-dimethyl-3-((3E,7E,11E)-3,7,12-trimethyl-14-(6...)
Affinity DataIC50:  0.220nMAssay Description:Inhibition of Candida albicans OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50094519((R)-1,1,1-Trifluoro-3-{(3-phenoxy-phenyl)-[3-(1,1,...)
Affinity DataIC50:  20nMAssay Description:Inhibition of CETP assessed as transfer of [3H]cholesterol esters from HDL to LDLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213696(3-((3E,7E)-11-((E)-4,8-dimethylnona-4,7-dienylthio...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50055641(2,2-dimethyl-3-((3E,7E,11E)-3,7,12-trimethyl-14-(6...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213692(2,2-dimethyl-3-((E)-3-methyl-7-((3E,8E)-4,8,12-tri...)
Affinity DataIC50:  50nMAssay Description:Inhibition of rat OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholesteryl ester transfer protein(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50094519((R)-1,1,1-Trifluoro-3-{(3-phenoxy-phenyl)-[3-(1,1,...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human CETP assessed as transfer of [3H]cholesterol esters from HDL to LDL in humna plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol synthase(Rattus norvegicus)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213691(1-((5S,6S,8aS)-6-hydroxy-5,8a-dimethyl-octahydrois...)
Affinity DataIC50:  700nMAssay Description:Inhibition of rat OSCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213683(CHEMBL218693 | carnosol)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of pancreatic lipaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213689((S)-2-((2E,8E)-deca-2,8-dienoylamino)-3-((S)-5-hyd...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of pancreatic lipaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50371232(CARNOSIC ACID)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of pancreatic lipaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLanosterol 14-alpha demethylase(Rattus norvegicus)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213698((1R,3aS,3bR,5aS,7S,9aS,9bS,11aR,E)-3,10-dihydroxy-...)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of rat liver LDMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213686(2-((2E,8E)-deca-2,8-dienoylamino)-3-(5-hydroxy-6-o...)
Affinity DataIC50:  1.20E+5nMAssay Description:Inhibition of pancreatic lipaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic triacylglycerol lipase(Homo sapiens (Human))
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50213694((R)-2-((2E,8E)-deca-2,8-dienoylamino)-3-((R)-5-hyd...)
Affinity DataIC50:  2.70E+5nMAssay Description:Inhibition of pancreatic lipaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(RABBIT)
Sinhgad College Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50118705(ABT-866 | CHEMBL326702 | Ethanesulfonic acid [3-(1...)
Affinity DataEC50:  60nMAssay Description:Agonist activity at rabbit urethra adrenergic alpha1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed