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Found 15 with Last Name = 'kaza' and Initial = 'sk'
TargetPotassium voltage-gated channel subfamily A member 1(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237249(CHEMBL4076021)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of recombinant rat Kv1.1 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin) expressed in HEK293 cells by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)4 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of recombinant rat Kv1.1 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 4(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of Kv1.4 (unknown origin) expressed in HEK293 cells by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM20461((6E)-N-[(4-hydroxy-3-methoxyphenyl)methyl]-8-methy...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50149890(CHEMBL9324 | tetraethylammonium)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)3/Kv1.2 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50:  5.70E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)2/Kv(1.2)2 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM10458(4-AP | 4-Aminopyridine 10 | CHEMBL284348 | DALFAMP...)
Affinity DataIC50:  8.90E+4nMAssay Description:Binding affinity towards 5-HT3 receptor in rat was evaluatedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50101817(Adalat | Adalat Cc | Afeditab Cr | BAY-A-1040 | CH...)
Affinity DataIC50:  9.60E+4nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetPotassium voltage-gated channel subfamily A member 1/2(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.1/Kv(1.2)3 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 2(Rattus norvegicus)
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.2(4) expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50004704((+)-cis-Diltiazem | (2S,3S)-5-(2-(dimethylamino)et...)
Affinity DataIC50:  1.44E+5nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 1(Homo sapiens (Human))
Dublin Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50131434(CHEMBL652 | FLECAINIDE | N-(piperidin-2-ylmethyl)-...)
Affinity DataIC50:  2.09E+5nMAssay Description:Inhibition of Kv1.1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed