Compile Data Set for Download or QSAR
maximum 50k data
Found 29 with Last Name = 'léger' and Initial = 'b'
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186073(CHEMBL210229 | N-(2-(dimethylamino)ethyl)-8-isopro...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186073(CHEMBL210229 | N-(2-(dimethylamino)ethyl)-8-isopro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186069(8-(4-methoxybenzyl)-2-(4,5-dihydro-1H-imidazol-2-y...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186085(8-(4-methoxybenzyl)-8,9-dihydrothiazolo[5,4-f]quin...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186086(8-benzyl-2-(4,5-dihydro-1H-imidazol-2-yl)thiazolo[...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186076(2-(4,5-dihydro-1H-imidazol-2-yl)-8-isopentylthiazo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186083(8-isobutyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186078(8-isopropyl-8,9-dihydrothiazolo[5,4-f]quinazoline-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186078(8-isopropyl-8,9-dihydrothiazolo[5,4-f]quinazoline-...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186076(2-(4,5-dihydro-1H-imidazol-2-yl)-8-isopentylthiazo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186075(8-benzyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2-c...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186077(8-ethyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2-ca...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186084(CHEMBL210474 | N-(2-(dimethylamino)ethyl)-8-ethyl-...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186077(8-ethyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2-ca...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186080(2-(4,5-dihydro-1H-imidazol-2-yl)-8-isobutylthiazol...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186082(8-ethyl-N-isopropyl-9-oxo-8,9-dihydrothiazolo[5,4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186072(CHEMBL378190 | N,8-diisopropyl-9-oxo-8,9-dihydroth...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186083(8-isobutyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186081(2-(4,5-dihydro-1H-imidazol-2-yl)-8-ethylthiazolo[5...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186079(8-isopentyl-8,9-dihydrothiazolo[5,4-f]quinazoline-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186071(2-(4,5-dihydro-1H-imidazol-2-yl)-8-isopropylthiazo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186074(8-propyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2-c...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186079(8-isopentyl-8,9-dihydrothiazolo[5,4-f]quinazoline-...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186074(8-propyl-8,9-dihydrothiazolo[5,4-f]quinazoline-2-c...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186081(2-(4,5-dihydro-1H-imidazol-2-yl)-8-ethylthiazolo[5...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186071(2-(4,5-dihydro-1H-imidazol-2-yl)-8-isopropylthiazo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186070(2-(4,5-dihydro-1H-imidazol-2-yl)-8-propylthiazolo[...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50186080(2-(4,5-dihydro-1H-imidazol-2-yl)-8-isobutylthiazol...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK5/p25 in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50186070(2-(4,5-dihydro-1H-imidazol-2-yl)-8-propylthiazolo[...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of CDK1/cyclinB in presence of 15 uM ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed