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Found 23 with Last Name = 'löscher' and Initial = 'w'
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122594(4,6-Dichloro-3-[(3-phenyl-ureido)-methyl]-1H-indol...)
Affinity DataKi:  14nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122590(4,6-Dichloro-3-(2,4-dioxo-3-phenyl-imidazolidin-1-...)
Affinity DataKi:  22nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122611(4,6-Dichloro-3-(2,4-dioxo-3-p-tolyl-imidazolidin-1...)
Affinity DataKi:  36nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122606(4,6-Dichloro-3-(2,4-dioxo-3-m-tolyl-imidazolidin-1...)
Affinity DataKi:  45nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122598(4,6-Dichloro-3-[3-(4-fluoro-phenyl)-2,4-dioxo-imid...)
Affinity DataKi:  53nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122602(3-[3-(3-Acetyl-phenyl)-2,4-dioxo-imidazolidin-1-yl...)
Affinity DataKi:  57nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122601(4,6-Dichloro-3-(2-oxo-3-phenyl-imidazolidin-1-ylme...)
Affinity DataKi:  58nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122591(4,6-dichloro-3-[({[(phenylsulfonyl)amino]carbonyl}...)
Affinity DataKi:  72nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122610(4,6-Dichloro-3-[3-(3,5-dichloro-phenyl)-2,4-dioxo-...)
Affinity DataKi:  80nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122608(4,6-Dichloro-3-[3-(3-chloro-phenyl)-2,4-dioxo-imid...)
Affinity DataKi:  85nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122593(4,6-Dichloro-3-[3-(4-methoxy-phenyl)-2,4-dioxo-imi...)
Affinity DataKi:  100nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122596(3-(Benzoylamino-methyl)-4,6-dichloro-1H-indole-2-c...)
Affinity DataKi:  120nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122600(4,6-Dichloro-3-[3-(4-chloro-phenyl)-2,4-dioxo-imid...)
Affinity DataKi:  120nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122605(4,6-Dichloro-3-(3-cyclohexyl-2,4-dioxo-imidazolidi...)
Affinity DataKi:  130nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122603(3-[3-(4-Acetyl-phenyl)-2,4-dioxo-imidazolidin-1-yl...)
Affinity DataKi:  150nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122609(4,6-Dichloro-3-(5-methyl-2,4-dioxo-3-phenyl-imidaz...)
Affinity DataKi:  310nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122595(4,6-Dichloro-3-(4-oxo-3-phenyl-2-thioxo-imidazolid...)
Affinity DataKi:  580nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122604(3-(Benzenesulfonylamino-methyl)-4,6-dichloro-1H-in...)
Affinity DataKi:  990nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122599(4,6-Dichloro-3-(3-ethyl-2,4-dioxo-imidazolidin-1-y...)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122592(4,6-Dichloro-3-(3-isopropyl-2,4-dioxo-imidazolidin...)
Affinity DataKi:  1.05E+3nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122597(4,6-Dichloro-3-(5-isopropyl-2,4-dioxo-3-phenyl-imi...)
Affinity DataKi:  1.10E+3nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50004960(4,6-Dichloro-1H-indole-2-carboxylic acid | CHEMBL3...)
Affinity DataKi:  2.90E+3nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor ionotropic, NMDA 1(Homo sapiens (Human))
Johannes Gutenberg-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50122607(3-(Benzylamino-methyl)-4,6-dichloro-1H-indole-2-ca...)
Affinity DataKi:  9.20E+4nMAssay Description:Tested for the affinity for the glycine binding site of the N-methyl-D-aspartate glutamate receptor using pig brain membranes in binding assay with [...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed