Compile Data Set for Download or QSAR
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Found 7 with Last Name = 'laethem' and Initial = 't'
TargetVoltage-dependent T-type calcium channel subunit alpha-1I(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392769(CHEMBL2151147)
Affinity DataIC50:  264nMAssay Description:Antagonist activity at Cav3.3 at -80 mV holding potential by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392766(CHEMBL2151144)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50338167((R)-2-(4-cyclopropylphenyl)-N-(1-(5-(2,2,2-trifluo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1I(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392769(CHEMBL2151147)
Affinity DataIC50:  1.20E+4nMAssay Description:Antagonist activity at Cav3.3 at -100 mV holding potential by whole cell patch clamp analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392769(CHEMBL2151147)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392767(CHEMBL2151145)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50392768(CHEMBL2151146)
Affinity DataIC50: >3.00E+4nMAssay Description:Displacement of [3S]MK499 from human ERG in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed