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Found 13 with Last Name = 'laine' and Initial = 'k'
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315227(CHEMBL1091204 | Isopropyl-3-chloro-5,6-dihydroxy-7...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315228(Butyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thioph...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315220((2-oxo-1,3-dioxol-4-yl)methyl 3-chloro-5,6-dihydro...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315230(CHEMBL1089504 | Methyl-3-chloro-5,6-dihydroxy-7-ni...)
Affinity DataKi:  2.20nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315221((2-amino-3-methylbutanoyloxy)methyl 3-chloro-5,6-d...)
Affinity DataKi:  6nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315229(CHEMBL1089505 | Propyl-3-chloro-5,6-dihydroxy-7-ni...)
Affinity DataKi:  9.20nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315226(Benzyl-3-chloro-5,6-dihydroxy-7-nitrobenzo[b]thiop...)
Affinity DataKi:  10.2nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315223(Butyryloxymethyl-3-chloro-5,6-dihydroxy-7-nitroben...)
Affinity DataKi:  10.6nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315222(1-(Butyryloxy)ethyl-3-chloro-5,6-dihydroxy-7-nitro...)
Affinity DataKi:  16.6nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315225(CHEMBL1089537 | Isobutyryloxymethyl-3-chloro-5,6-d...)
Affinity DataKi:  17nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCatechol O-methyltransferase(Homo sapiens (Human))
University Of Eastern Finland

Curated by ChEMBL
LigandPNGBDBM50315224(1-(Isobutyryloxy)ethyl-3-chloro-5,6-dihydroxy-7-ni...)
Affinity DataKi:  17nMAssay Description:Inhibition of human recombinant COMT by microplate screening assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Rattus norvegicus)
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50250177(((2R,3S,4S,5R,6R)-3,4,5,6-tetrahydroxytetrahydro-2...)
Affinity DataIC50:  710nMAssay Description:Inhibition of GluT1-mediated [14C]D-glucose uptake in Wistar rat brain by perfusion techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Rattus norvegicus)
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50250141(((2R,3S,4S,5R,6R)-3,4,5,6-tetrahydroxytetrahydro-2...)
Affinity DataIC50:  3.29E+4nMAssay Description:Inhibition of GluT1-mediated [14C]D-glucose uptake in Wistar rat brain by perfusion techniqueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed