Affinity DataEC50: 794nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 5.01E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 2.51E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 2.51E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 7.94E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 158nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 2.00E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 398nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: >3.16E+4nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 501nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 100nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.58E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 3.98E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 1.26E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
Affinity DataEC50: 794nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 251nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 126nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 501nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 3.16E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 631nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 631nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 794nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.58E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 2.51E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 2.00E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Positive modulation of GluR1More data for this Ligand-Target Pair
Affinity DataEC50: 1.00E+3nMAssay Description:Modulatory activity at GluA2 receptor LBDMore data for this Ligand-Target Pair