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Found 750 with Last Name = 'lan' and Initial = 'x'
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM86211(CAS_52809-07-1 | NSC_40539 | Quisqualate)
Affinity DataKi:  0.0300nMMore data for this Ligand-Target Pair
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556826(CHEMBL4745863)
Affinity DataKi:  0.220nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556827(CHEMBL4748838)
Affinity DataKi:  0.25nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50002371(2-aminopentanedioic acidglutamic acid | CHEMBL2763...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556825(CHEMBL4787784)
Affinity DataKi:  0.460nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by PDSP Ki Database
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  0.560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556828(CHEMBL4798771)
Affinity DataKi:  0.600nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50089896(4-(Amino-carboxy-methyl)-3-methyl-benzoic acid((+)...)
Affinity DataKi:  1.18nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Johnson & Johnson Pharmaceutical Research And Development

Curated by PDSP Ki Database
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  1.26nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50163606(1-(3,4-Dihydro-2H-1-oxa-9-aza-anthracen-6-yl)-2-ph...)
Affinity DataKi:  1.35nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50231744(CHEMBL399160 | NPS 2390 | quinoxaline-2-carboxylic...)
Affinity DataKi:  1.36nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50030628((S)-4C3HPG | 4-(Amino-carboxy-methyl)-2-hydroxy-be...)
Affinity DataKi:  1.65nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM86212(1S, 3R-ACPD | CAS_104766 | NSC_104766)
Affinity DataKi:  1.92nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHrh3 protein(RAT)
Johnson & Johnson Pharmaceutical Research And Development

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  3.98nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50030629((R,S)-4-Carboxy-3-hydroxyphenylglycine | (S)-4CPG ...)
Affinity DataKi:  4.51nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556824(CHEMBL4746142)
Affinity DataKi:  5.10nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology

Curated by ChEMBL
LigandPNGBDBM50556829(CHEMBL4743589)
Affinity DataKi:  5.60nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  8.30nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  8.90nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50212323((3aS,6aS)-5-methylene-6a-(naphthalen-2-ylmethyl)-h...)
Affinity DataKi:  11.2nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50163631(1-Methyl-4-piperidin-4-ylidene-1,4-dihydro-1,5,7a-...)
Affinity DataKi:  12nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209684(CHEMBL390718 | cis-(+)-7,8-dimethoxy-3-[4-(2-methy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50163629(CHEMBL539843 | spiro[6,11-dihydro-5H-benzo[d]imida...)
Affinity DataKi:  19nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50163630(1-Methyl-4-piperidin-4-ylidene-1,4,8,9-tetrahydro-...)
Affinity DataKi:  22nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM22876(CHEMBL998 | Claritin | Loratadine | Sch 29851 | US...)
Affinity DataKi:  37nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM22890(2-(2-{4-[(4-chlorophenyl)(phenyl)methyl]piperazin-...)
Affinity DataKi:  50nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetTransporter(Rattus norvegicus)
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]nisoxetine from rat NETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  72nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]pyrilamine from human cloned histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development

Curated by PDSP Ki Database
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)
Affinity DataKi:  79.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse

Curated by PDSP Ki Database
LigandPNGBDBM50030630((RS)-1-aminoindan-1,5-dicarboxylic acid | 1-Amino-...)
Affinity DataKi:  98.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  117nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50146518((3R,3aS)-3-{4-[3-(4-Fluoro-phenyl)-2-methyl-allyl]...)
Affinity DataKi:  125nMAssay Description:Displacement of [3H]prazosin from human cloned alpha-1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50209685(CHEMBL226636 | cis-(+)-7,8-dimethoxy-3-[4-(3-(4-fl...)
Affinity DataKi:  162nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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