TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology
Curated by ChEMBL
Huazhong University Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 0.220nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology
Curated by ChEMBL
Huazhong University Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology
Curated by ChEMBL
Huazhong University Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology
Curated by ChEMBL
Huazhong University Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetHrh3 protein(RAT)
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetHrh3 protein(RAT)
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology
Curated by ChEMBL
Huazhong University Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 5.10nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
TargetApelin receptor(Homo sapiens (Human))
Huazhong University Of Science & Technology
Curated by ChEMBL
Huazhong University Of Science & Technology
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [Glp65, Nle75, Tyr77][125I]-apelin13 from human APJ receptor expressed in HEK293 cells incubated for 1 hr by gamma counting based rad...More data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.30nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Displacement of [3H]paroxetine from human cloned 5HTT receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Binding affinity for H1 histamine receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Displacement of [3H]nisoxetine from rat NETMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 72nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic Alpha-2C receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H1 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Johnson & Johnson Pharmaceutical Research & Development
Curated by ChEMBL
Affinity DataKi: 74nMAssay Description:Displacement of [3H]pyrilamine from human cloned histamine H1 receptorMore data for this Ligand-Target Pair
TargetHistamine H4 receptor(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
Johnson & Johnson Pharmaceutical Research And Development
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 1(RAT)
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Johnson And Johnson Pharmaceutical Research And Development, Beerse
Curated by PDSP Ki Database
Affinity DataKi: 117nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 117nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha2A receptor transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Displacement of [3H]prazosin from human cloned alpha-1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 162nMAssay Description:Displacement of [3H]rawolscine from human cloned adrenergic alpha-2B receptor transfected in CHO cellsMore data for this Ligand-Target Pair