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Found 64 with Last Name = 'lanba' and Initial = 'a'
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195581((2R,3R)-2-(3-ethynylphenyl)-1-(3-(4-(2-morpholinop...)
Affinity DataIC50:  5nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195574((R)-(2-phenylpiperidin-1-yl)(3-(4-(pyridin-3-yl)ph...)
Affinity DataIC50:  5nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195575((R)-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H-1...)
Affinity DataIC50:  5nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195572((R)-N,N-dimethyl-4'-(2-(2-phenylpiperidine-1-c...)
Affinity DataIC50: <5nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195571((R)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...)
Affinity DataIC50: <5nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195570((S)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...)
Affinity DataIC50: <5nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195580((2R,3R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...)
Affinity DataIC50:  6nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195573((R)-4'-(1-(2-phenylpiperidine-1-carbonyl)-1H-1...)
Affinity DataIC50:  7nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195575((R)-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H-1...)
Affinity DataIC50:  7nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195578((2R, 4R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)pheny...)
Affinity DataIC50:  11nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195572((R)-N,N-dimethyl-4'-(2-(2-phenylpiperidine-1-c...)
Affinity DataIC50:  21nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195574((R)-(2-phenylpiperidin-1-yl)(3-(4-(pyridin-3-yl)ph...)
Affinity DataIC50:  36nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195573((R)-4'-(1-(2-phenylpiperidine-1-carbonyl)-1H-1...)
Affinity DataIC50:  48nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195571((R)-4'-(2-(2-phenylpiperidine-1-carbonyl)-2H-1...)
Affinity DataIC50:  59nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149290(CHEMBL3771175)
Affinity DataIC50:  110nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149291(CHEMBL3770609)
Affinity DataIC50:  110nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149290(CHEMBL3771175)
Affinity DataIC50:  110nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149291(CHEMBL3770609)
Affinity DataIC50:  110nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  120nMAssay Description:Inhibition of NaCT in rat hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Rattus norvegicus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  126nMAssay Description:Inhibition of NaCT in rat hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149289(CHEMBL3770497)
Affinity DataIC50:  190nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149289(CHEMBL3770497)
Affinity DataIC50:  200nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  210nMAssay Description:Inhibition of NaCT in mouse hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Mus musculus)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  214nMAssay Description:Inhibition of NaCT in mouse hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149291(CHEMBL3770609)
Affinity DataIC50:  316nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149293(CHEMBL3770675)
Affinity DataIC50:  316nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149291(CHEMBL3770609)
Affinity DataIC50:  330nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149293(CHEMBL3770675)
Affinity DataIC50:  330nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50:  501nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149294(CHEMBL3769578)
Affinity DataIC50:  501nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  501nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  510nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149236(CHEMBL3770370)
Affinity DataIC50:  650nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149236(CHEMBL3770370)
Affinity DataIC50:  650nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195576(cis-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl)-1H...)
Affinity DataIC50:  710nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  740nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149215(CHEMBL3769514)
Affinity DataIC50:  794nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  794nMAssay Description:Inhibition of NaCT in human hepatocytes assessed as [14C]-citrate uptake after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149215(CHEMBL3769514)
Affinity DataIC50:  800nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195579((2S,3S)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...)
Affinity DataIC50:  1.10E+3nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149233(CHEMBL3769911)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149233(CHEMBL3769911)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149247(CHEMBL3769766)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149247(CHEMBL3769766)
Affinity DataIC50:  3.37E+3nMAssay Description:Inhibition of NaCT (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLiver carboxylesterase 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195578((2R, 4R)-1-(3-(4-(2-morpholinopyrimidin-5-yl)pheny...)
Affinity DataIC50:  3.70E+3nMpH: 7.5Assay Description:For determination of IC50 values for CES1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of 25...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysophospholipase-like protein 1(Homo sapiens (Human))
Pfizer

LigandPNGBDBM195577((2S,4S)-1-(3-(4-(2-morpholinopyrimidin-5-yl)phenyl...)
Affinity DataIC50:  6.50E+3nMpH: 7.5Assay Description:For determination of IC50 values for LYPLAL1 inhibitors, the reactions were carried out in 1.5 mL microcentrifuge tubes in a total reaction volume of...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of NaDC1 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 2(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of NaDC1 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of NaDC3 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 13 member 3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50149244(CHEMBL3771118)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibition of NaDC3 (unknown origin) expressed in HEK293 cells assessed as inhibition of [14C]citrate uptake by microbeta plate reader analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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