Compile Data Set for Download or QSAR
maximum 50k data
Found 154 with Last Name = 'lawson' and Initial = 'ja'
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014100(2-(1-{[1-{2-Hydroxy-1-isobutyl-5-methyl-4-[2-methy...)
Affinity DataIC50:  0.260nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014102(Boc-Pro-Phe-N(Me) His-Leu[CHOHCH2]Val-Ile-THAM Ami...)
Affinity DataIC50:  0.260nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011341(2-Amino-5-[2-(1-{[1-[1-cyclohexylmethyl-2-hydroxy-...)
Affinity DataIC50:  0.280nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011339(2-Amino-5-[2-(1-{[1-(1-cyclohexylmethyl-2-hydroxy-...)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011347(5-[2-{[2-(3-Amino-3-methyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  0.290nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50406474(CHEMBL2028945)
Affinity DataIC50:  0.310nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011342(2-Amino-5-[2-(1-{[1-(1-cyclohexylmethyl-2-hydroxy-...)
Affinity DataIC50:  0.320nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014106(CHEMBL429882 | N-[[[2-Hydroxy-1,1-bis(hydroxymethy...)
Affinity DataIC50:  0.330nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014105(2-(1-{[1-{2-Hydroxy-1-isobutyl-5-methyl-4-[2-methy...)
Affinity DataIC50:  0.330nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011337(5-[2-{[2-(3-Amino-3-methyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  0.410nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011348(5-[2-{[2-(3-Amino-3-methyl-butyrylamino)-3-phenyl-...)
Affinity DataIC50:  0.430nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011345(CHEMBL3143483 | Phosphoric acid mono-{4-[2-(1-{[1-...)
Affinity DataIC50:  0.450nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014099(CHEMBL414795 | N-[(D-Glucosylamino)carbonyl]-Pro-P...)
Affinity DataIC50:  0.490nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014104(CHEMBL410067 | N-[[[2-Hydroxy-1,1-bis(hydroxymethy...)
Affinity DataIC50:  0.580nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011343(CHEMBL3143477 | Sodium; 2-{[7-(1-{[1-(2-hydroxy-1-...)
Affinity DataIC50:  0.660nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014101(CHEMBL265833 | N-[4,5-Dihydro-4,4-bis(hydroxymethy...)
Affinity DataIC50:  1.10nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Rattus norvegicus)
Upjohn

Curated by ChEMBL
LigandPNGBDBM50014103(CHEMBL263257 | N-[(D-Glucosylamino)carbonyl]-Pro-P...)
Affinity DataIC50:  1.10nMAssay Description:Tested invitro for inhibitory activity against plasma renin in rat modelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011346(CHEMBL3143482 | Sodium; 2-{[7-(1-{[1-(2-hydroxy-1-...)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50011350(CHEMBL3143484 | Phosphoric acid mono-{2-[2-(1-{[1-...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50024214(Boc-alpha-MePro-Phe-His-Leu si[CHOHCH2]Val-Ile-Amp...)
Affinity DataIC50:  1.60nMAssay Description:In vitro inhibition against human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50406476(CHEMBL2028948)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50406473(CHEMBL2028947)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50367481(CHEMBL1237141 | CHEMBL3143428)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition against hog renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367061(NALORPHINE | NALORPHINE HYDROCHLORIDE)
Affinity DataIC50:  2nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50406475(CHEMBL2028946)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497135(CHEMBL3275470)
Affinity DataIC50:  3.40nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50024212(2-{1-[1-[1-(1-Hydroxy-2-{2-methyl-1-[(pyridin-2-yl...)
Affinity DataIC50:  3.5nMAssay Description:In vitro inhibition against human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497128(CHEMBL3275472)
Affinity DataIC50:  4.20nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50367061(NALORPHINE | NALORPHINE HYDROCHLORIDE)
Affinity DataIC50:  6nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in presence of NaClMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497127(CHEMBL3275471)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497127(CHEMBL3275471)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in presence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497134(CHEMBL3275464)
Affinity DataIC50:  16nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497126(CHEMBL3275469)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50024161((1-{1-[1-(1-Hydroxy-2-{2-methyl-1-[(pyridin-2-ylme...)
Affinity DataIC50:  24nMAssay Description:In vitro inhibition against human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497134(CHEMBL3275464)
Affinity DataIC50:  25nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in presence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50367718(CHEMBL3037868)
Affinity DataIC50:  26nMAssay Description:In vitro inhibitory activity against renin from lyophilized human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497131(CHEMBL3275463)
Affinity DataIC50:  27nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497122(CHEMBL3275461)
Affinity DataIC50:  28nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497123(CHEMBL3275467)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50024213(2-(1-{1-[1-(1-Hydroxy-2-{2-methyl-1-[(pyridin-2-yl...)
Affinity DataIC50:  36nMAssay Description:In vitro inhibition against human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497132(CHEMBL3275465)
Affinity DataIC50:  37nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497121(CHEMBL3272387)
Affinity DataIC50:  38nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50367482(CHEMBL1237142 | CHEMBL3144387)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition against hog renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50024215(2-[1-(2-(1H-Imidazol-4-yl)-1-{3-methyl-1-[(2-methy...)
Affinity DataIC50:  43nMAssay Description:In vitro inhibition against human plasma renin.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497123(CHEMBL3275467)
Affinity DataIC50:  45nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in presence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Upjohn

Curated by ChEMBL
LigandPNGBDBM50367714(CHEMBL1790111)
Affinity DataIC50:  49nMAssay Description:In vitro inhibitory activity against renin from lyophilized human plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497125(CHEMBL3275468)
Affinity DataIC50:  51nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497124(CHEMBL3275462)
Affinity DataIC50:  60nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in absence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type/Kappa-type/Mu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50497122(CHEMBL3275461)
Affinity DataIC50:  62nMAssay Description:Displacement of [3H]-naloxone from rat opioid receptor after 30 mins by liquid scintillation counting analysis in presence of NaClMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 154 total ) | Next | Last >>
Jump to: