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Found 27 with Last Name = 'leal' and Initial = 'j'
LigandPNGBDBM50080742((S)-2-[(5-{[Benzyl-(5-fluoro-pyridin-3-yl)-amino]-...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080765((S)-2-({5-[(Cyclohexylmethyl-pyridin-3-yl-amino)-m...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080764((S)-2-({5-[(Benzyl-pyridin-3-yl-amino)-methyl]-2'-...)
Affinity DataIC50:  0.100nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080748((S)-2-[(5-{[(3,5-Difluoro-benzyl)-thiazol-5-ylmeth...)
Affinity DataIC50:  0.200nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080743((S)-2-({5-[(Benzyl-thiazol-5-ylmethyl-amino)-methy...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067563((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-biphen...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080750((S)-2-({5-[(Benzyl-pyrimidin-5-yl-amino)-methyl]-2...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50067581((S)-2-{[2'-Methyl-5-(pyridin-3-ylaminomethyl)-biph...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080747((S)-2-[(5-{[(3,5-Difluoro-benzyl)-phenyl-amino]-me...)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080759((S)-2-{[2'-Methyl-4-phenethyl-5-(pyridin-3-yloxyme...)
Affinity DataIC50:  0.5nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080744((S)-2-({5-[(Benzyl-pyrazin-2-yl-amino)-methyl]-2'-...)
Affinity DataIC50:  0.800nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080762((S)-2-{[4-Benzyl-2'-methyl-5-(pyridin-3-yloxymethy...)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080763((S)-2-[(5-{[(3,5-Difluoro-benzyl)-pyridin-3-yl-ami...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080745((S)-2-({5-[(Benzyl-phenyl-amino)-methyl]-2'-methyl...)
Affinity DataIC50:  1.40nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080761((S)-2-{[2'-Methyl-4-pentyl-5-(pyridin-3-yloxymethy...)
Affinity DataIC50:  2nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080760((S)-2-{[4-Ethyl-2'-methyl-5-(pyridin-3-yloxymethyl...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080752((S)-2-({5-[(Benzyl-thiazol-2-ylmethyl-amino)-methy...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080751((S)-2-({5-[(Benzenesulfonyl-pyridin-3-yl-amino)-me...)
Affinity DataIC50:  7nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080749((S)-2-{[4-Butyl-2'-methyl-5-(pyridin-3-yloxymethyl...)
Affinity DataIC50:  11nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080756((S)-2-{[4-Cyclohexylmethyl-2'-methyl-5-(pyridin-3-...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080753((S)-2-({5-[(Benzyl-thiazol-4-ylmethyl-amino)-methy...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080755((S)-2-{[4-Isobutyl-2'-methyl-5-(pyridin-3-yloxymet...)
Affinity DataIC50:  29nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080754((S)-2-({2'-Methyl-5-[(phenylacetyl-pyridin-3-yl-am...)
Affinity DataIC50:  39nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080757((S)-2-({5-[(Benzoyl-pyridin-3-yl-amino)-methyl]-2'...)
Affinity DataIC50:  53nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080758((S)-2-{[3'',5''-Dichloro-2-methyl-5'-(pyridin-3-yl...)
Affinity DataIC50:  95nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080746((S)-2-{[2,4''-Dimethyl-5'-(pyridin-3-yloxymethyl)-...)
Affinity DataIC50:  370nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50080766((S)-2-{[2'-Methyl-5-(pyridin-3-yloxymethyl)-4-thio...)
Affinity DataIC50:  510nMAssay Description:In vitro inhibition of farnesyltransferase purified from bovine brain using scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed