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Found 38 with Last Name = 'lebedev' and Initial = 'r'
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212403((1R,2R)-2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,...)
Affinity DataEC50:  2.30nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212273(3-(3-(1,4,4,6-tetramethyl-2-oxo-1,2,3,4-tetrahydro...)
Affinity DataEC50:  24.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212407((Z)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  39.1nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212408(2-(3-(1,4,4,6-tetramethyl-2-oxo-1,2,3,4-tetrahydro...)
Affinity DataEC50:  144nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212409((1R,2R)-2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,...)
Affinity DataEC50:  10nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212414(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  760nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212404(2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  19.2nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212415(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  36.5nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212412(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  361nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212418(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  7.20nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212417(3-(4-(trifluoromethoxy)-3-(4,4,6-trimethyl-2-oxo-1...)
Affinity DataEC50:  1.40nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212274(5-((3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetra...)
Affinity DataEC50:  0.900nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212419(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212411(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  37.7nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212277((E)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212413((1S,2S)-2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,...)
Affinity DataEC50:  361nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212423(3-(3-(1,4,4,6-tetramethyl-2-oxo-1,2,3,4-tetrahydro...)
Affinity DataEC50:  45.9nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212410(4-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  527nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212416((1S,2S)-2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,...)
Affinity DataEC50:  198nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212406(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  3.40nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212422(2-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  116nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212426(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  27.9nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212425(2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  208nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212427(2-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  5nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212264(3-(3-(4-ethyl-2,2,7-trimethyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  61.2nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212268(3-(3-(5-ethyl-4-oxo-2,3,4,5-tetrahydro-1H-cyclopen...)
Affinity DataEC50:  96.6nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212269((E)-3-(5-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  1.20E+3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212271(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  16.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212276(3-(3-(4-ethyl-2,2,7-trimethyl-3-oxo-3,4-dihydro-2H...)
Affinity DataEC50:  173nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212281(3-(5-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212283((E)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  67.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212272(3-(3-(5-ethyl-8-methyl-4-oxo-2,3,4,5-tetrahydro-1H...)
Affinity DataEC50:  1.60E+3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212266(3-(4-(trifluoromethoxy)-3-(4,4,6-trimethyl-2-oxo-1...)
Affinity DataEC50:  2.10nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212275(3-(4-(trifluoromethoxy)-3-(4,4,6-trimethyl-2-oxo-1...)
Affinity DataEC50:  1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212267(3-(3-(1-isopropyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  18.3nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212274(5-((3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetra...)
Affinity DataEC50:  0.900nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212277((E)-3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-te...)
Affinity DataEC50:  1.80nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-alpha(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50212405(3-(3-(1-ethyl-4,4,6-trimethyl-2-oxo-1,2,3,4-tetrah...)
Affinity DataEC50:  70.2nMAssay Description:Activity at RXRalpha by GAL4DNA cotransfection assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed