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Found 108 with Last Name = 'lefrançois' and Initial = 'd'
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093978(2-(4-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  0.810nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093997(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093996(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094000(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093987(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.30nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093997(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093999(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093985(2-(6-Carboxy-4H-benzo[1,3]dioxin-8-ylmethyl)-4-(6-...)
Affinity DataIC50:  2.5nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093993(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  2.60nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093996(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093995(2-(2-Carboxymethoxy-cyclohexylmethyl)-4-(6-chloro-...)
Affinity DataIC50:  3.20nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093984(2-(2-Carboxymethoxy-benzyl)-4-(6-chloro-benzo[1,3]...)
Affinity DataIC50:  3.30nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093980(2-Adamantan-1-ylmethyl-4-(6-chloro-benzo[1,3]dioxo...)
Affinity DataIC50:  3.40nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094004(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  3.40nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093993(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  3.60nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093988(2-(2-Carboxymethoxy-4-methoxy-benzyl)-4-(6-chloro-...)
Affinity DataIC50:  4nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093986(2-(2-Carboxymethoxy-benzyl)-4-(6-chloro-benzo[1,3]...)
Affinity DataIC50:  4.60nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094004(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  4.70nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094003(2-(4-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  4.90nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093980(2-Adamantan-1-ylmethyl-4-(6-chloro-benzo[1,3]dioxo...)
Affinity DataIC50:  4.90nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094002(2-(3-Carboxy-benzyl)-4-(6-chloro-benzo[1,3]dioxol-...)
Affinity DataIC50:  6.20nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093990(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  6.30nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093981(2-(2-Carboxymethoxy-4-methoxy-benzyl)-4-(6-chloro-...)
Affinity DataIC50:  8.60nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094001(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3,5-di...)
Affinity DataIC50:  9.70nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093987(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  9.80nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094000(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  9.90nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093998(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3-chlo...)
Affinity DataIC50:  11nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093994(2-(4-Carboxy-benzyl)-4-(6-chloro-benzo[1,3]dioxol-...)
Affinity DataIC50:  11nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093981(2-(2-Carboxymethoxy-4-methoxy-benzyl)-4-(6-chloro-...)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093992(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(2-ethy...)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093999(2-(3-Carboxy-cyclohexylmethyl)-4-(6-chloro-benzo[1...)
Affinity DataIC50:  15nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093998(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3-chlo...)
Affinity DataIC50:  17nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093990(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-cyclohe...)
Affinity DataIC50:  18nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50089716(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3-meth...)
Affinity DataIC50:  18nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50089716(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3-meth...)
Affinity DataIC50:  18nMAssay Description:In vitro inhibition of endothelin binding to endothelin A receptor in rat heart ventricles was measured using a 125-I labelled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093995(2-(2-Carboxymethoxy-cyclohexylmethyl)-4-(6-chloro-...)
Affinity DataIC50:  21nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093991(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3,4-di...)
Affinity DataIC50:  26nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50089721(4-Benzo[1,3]dioxol-5-ylmethyl-2-(3-methoxy-benzyl)...)
Affinity DataIC50:  28nMAssay Description:In vitro inhibition of endothelin binding to endothelin A receptor in rat heart ventricles was measured using a 125-I labelled ET-1 competition assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094001(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3,5-di...)
Affinity DataIC50:  28nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093986(2-(2-Carboxymethoxy-benzyl)-4-(6-chloro-benzo[1,3]...)
Affinity DataIC50:  28nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093992(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(2-ethy...)
Affinity DataIC50:  31nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093991(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3,4-di...)
Affinity DataIC50:  34nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50089716(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3-meth...)
Affinity DataIC50:  34nMAssay Description:In vitro inhibition of [125-I] labelled ET-1 endothelin binding to Endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50089716(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-(3-meth...)
Affinity DataIC50:  34nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50089721(4-Benzo[1,3]dioxol-5-ylmethyl-2-(3-methoxy-benzyl)...)
Affinity DataIC50:  40nMAssay Description:In vitro inhibition of [125-I] labelled ET-1 endothelin binding to Endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093985(2-(6-Carboxy-4H-benzo[1,3]dioxin-8-ylmethyl)-4-(6-...)
Affinity DataIC50:  44nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093984(2-(2-Carboxymethoxy-benzyl)-4-(6-chloro-benzo[1,3]...)
Affinity DataIC50:  59nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093979(4-(6-Chloro-benzo[1,3]dioxol-5-ylmethyl)-2-[1,3]di...)
Affinity DataIC50:  70nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-1 receptor(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50093989(5-[5-Carboxy-4-(6-chloro-benzo[1,3]dioxol-5-ylmeth...)
Affinity DataIC50:  79nMAssay Description:In vitro binding affinity to endothelin A receptor in rat heart ventriclesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin receptor type B(RAT)
Hoechst Marion Roussel

Curated by ChEMBL
LigandPNGBDBM50094002(2-(3-Carboxy-benzyl)-4-(6-chloro-benzo[1,3]dioxol-...)
Affinity DataIC50:  89nMAssay Description:In vitro binding affinity to endothelin B receptor in rat cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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