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Found 63 with Last Name = 'legiec' and Initial = 'ie'
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185143((+/-)-2-(cis-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-ox...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185145((+/-)-2-(cis-5-(4-(5-(4-((S)-3,3-difluorocyclopent...)
Affinity DataIC50:  0.800nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185147((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-3-fluorophenyl...)
Affinity DataIC50:  2nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185146((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-2-fluorophenyl...)
Affinity DataIC50:  2.70nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  2.90nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185149((+/-)-2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxad...)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185144((+/-)-3-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxad...)
Affinity DataIC50:  4.5nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185142((+/-)-3-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  5.70nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185150((+/-)-2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  8nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  13nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  13nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185145((+/-)-2-(cis-5-(4-(5-(4-((S)-3,3-difluorocyclopent...)
Affinity DataIC50:  16nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185151((+/-)-trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadi...)
Affinity DataIC50:  17nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  19nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185143((+/-)-2-(cis-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-ox...)
Affinity DataIC50:  20nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185147((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-3-fluorophenyl...)
Affinity DataIC50:  30nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185144((+/-)-3-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxad...)
Affinity DataIC50:  30nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185146((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-2-fluorophenyl...)
Affinity DataIC50:  60nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 1(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185148((+/-)-cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiaz...)
Affinity DataIC50:  75nMAssay Description:Displacement of [33P]S1P from S1P1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185142((+/-)-3-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  80nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185150((+/-)-2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  100nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185151((+/-)-trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadi...)
Affinity DataIC50:  180nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185149((+/-)-2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxad...)
Affinity DataIC50:  200nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185151((+/-)-trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadi...)
Affinity DataIC50:  300nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185143((+/-)-2-(cis-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-ox...)
Affinity DataIC50:  350nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185144((+/-)-3-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxad...)
Affinity DataIC50:  540nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  570nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  570nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185142((+/-)-3-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  630nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185150((+/-)-2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  700nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185145((+/-)-2-(cis-5-(4-(5-(4-((S)-3,3-difluorocyclopent...)
Affinity DataIC50:  720nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185149((+/-)-2-(cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxad...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185148((+/-)-cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiaz...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 5(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185148((+/-)-cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiaz...)
Affinity DataIC50:  1.28E+3nMAssay Description:Displacement of [33P]S1P from S1P5 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185146((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-2-fluorophenyl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185143((+/-)-2-(cis-5-(4-(5-(4-cyclohexylphenyl)-1,2,4-ox...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 4(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185147((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-3-fluorophenyl...)
Affinity DataIC50:  2.10E+3nMAssay Description:Displacement of [33P]S1P from S1P4 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185145((+/-)-2-(cis-5-(4-(5-(4-((S)-3,3-difluorocyclopent...)
Affinity DataIC50:  2.20E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185142((+/-)-3-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50:  6.70E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185147((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-3-fluorophenyl...)
Affinity DataIC50:  7.60E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185141((+/-)-2-(cis-5-(4-(5-(4-((R)-3,3-difluorocyclopent...)
Affinity DataIC50:  7.80E+3nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185150((+/-)-2-(trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-ox...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185148((+/-)-cis-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadiaz...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185151((+/-)-trans-5-(4-(5-(4-isobutylphenyl)-1,2,4-oxadi...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [33P]S1P from S1P2 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine 1-phosphate receptor 3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185146((+/-)-2-(cis-5-(4-(5-(4-cyclopentyl-2-fluorophenyl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [33P]S1P from S1P3 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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