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Found 8 with Last Name = 'lehane' and Initial = 'am'
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM81939(CAS_52-53-9 | NSC_62969 | VERAPAMIL)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM35938(1-(p-chlorophenyl)-1-(2-pyridyl)-3-N,N-dimethylpro...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50020157(CHEMBL3288457)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50020159(CHEMBL3286418)
Affinity DataIC50:  6.60E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM71542((4-amino-1-methyl-butyl)-(6-methoxy-8-quinolyl)ami...)
Affinity DataIC50:  6.80E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50017696((2-dimethylamino-2-methyl)ethyl-N-dibenzoparathiaz...)
Affinity DataIC50:  8.50E+4nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50020160(CHEMBL3288467)
Affinity DataIC50:  1.80E+5nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetChloroquine resistance transporter(Plasmodium falciparum)
Australian National University

Curated by ChEMBL
LigandPNGBDBM50020154(CHEMBL3288452)
Affinity DataIC50:  3.21E+5nMAssay Description:Inhibition of chloroquine-resistant Plasmodium falciparum Dd2 CRT expressed in Xenopus laevis oocytes plasma membrane assessed as reduction of [3H]-c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed