TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.300nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.5nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]ABP688 from human mGluR5 receptor expressed in L (tk-) cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]ABP688 from mGluR5 in rat brain membraneMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 2.60nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]M-MPEP from human mGluR5 receptor expressed in L (tk-) cellsMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 4.20nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 6.70nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]ABP688 from human mGluR5 receptor expressed in L (tk-) cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]ABP688 from mGluR5 in rat brain membraneMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 14nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 18nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]ABP688 from mGluR5 in rat brain membraneMore data for this Ligand-Target Pair
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of endothelin-converting enzyme in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:In vitro displacement of [3H]-LY 278584 from rat cerebral cortex 5-hydroxytryptamine 3 receptorMore data for this Ligand-Target Pair
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Inhibition of endothelin-converting enzyme in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Novartis Institutes For Biomedical Research
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]ABP688 from human mGluR5 receptor expressed in L (tk-) cellsMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 26nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 29nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Inhibition of VKORC1 in rat liver microsomes in presence of 0.003 to 0.2 mM vitamin KMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 36nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 38nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Novartis Institute For Medical Sciences
Curated by ChEMBL
Novartis Institute For Medical Sciences
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:In vitro binding affinity towards Tachykinin receptor 1 by measuring its ability to displace [3H]SP (0.6 nM) binding to membranes from Cos-7 cells tr...More data for this Ligand-Target Pair
TargetVitamin K epoxide reductase complex subunit 1(Rattus norvegicus (Rat))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Inhibition of neutral endopeptidase in human umbilical vein endothelial cellsMore data for this Ligand-Target Pair