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Found 1031 with Last Name = 'li' and Initial = 'mm'
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50005397(CHEMBL2206684)
Affinity DataKi:  0nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402366(CHEMBL2206696)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50005398(CHEMBL2206694)
Affinity DataKi:  0.00100nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402373(CHEMBL2206691)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402378(CHEMBL2206685)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402361(CHEMBL2206680)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402360(CHEMBL2206681)
Affinity DataKi:  0.00200nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402374(CHEMBL2206690)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402372(CHEMBL2206692)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402371(CHEMBL2206693)
Affinity DataKi:  0.00300nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402362(CHEMBL2206700)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402363(CHEMBL2206699)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402375(CHEMBL2206689)
Affinity DataKi:  0.00400nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402370(CHEMBL2206683)
Affinity DataKi:  0.00600nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402367(CHEMBL2206695)
Affinity DataKi:  0.00700nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402376(CHEMBL2206688)
Affinity DataKi:  0.00800nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402364(CHEMBL2206698)
Affinity DataKi:  0.0110nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402365(CHEMBL2206697)
Affinity DataKi:  0.0120nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402377(CHEMBL2206687)
Affinity DataKi:  0.0330nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402379(CHEMBL2206686)
Affinity DataKi:  0.296nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402368(CHEMBL2206682)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase plasminogen activator surface receptor(Homo sapiens (Human))
National Research Center

Curated by ChEMBL
LigandPNGBDBM50402369(CHEMBL1652555)
Affinity DataKi:  20.8nMAssay Description:Binding affinity to uPARMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50398211(CHEMBL2181036)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]chrysamine G from fibrillar amyloid beta (1 to 40) (unknown origin) after 1 hr by liquid scintillation spectrophotometric analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50002834(CHEMBL3233658)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]chrysamine G from fibrillar amyloid beta (1 to 40) (unknown origin) after 1 hr by liquid scintillation spectrophotometric analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50002835(CHEMBL3233659)
Affinity DataKi:  56nMAssay Description:Displacement of [3H]chrysamine G from fibrillar amyloid beta (1 to 40) (unknown origin) after 1 hr by liquid scintillation spectrophotometric analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50002836(CHEMBL3233660)
Affinity DataKi:  84nMAssay Description:Displacement of [3H]chrysamine G from fibrillar amyloid beta (1 to 40) (unknown origin) after 1 hr by liquid scintillation spectrophotometric analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmyloid-beta precursor protein(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50002833(CHEMBL3233657)
Affinity DataKi:  244nMAssay Description:Displacement of [3H]chrysamine G from fibrillar amyloid beta (1 to 40) (unknown origin) after 1 hr by liquid scintillation spectrophotometric analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein phosphatase non-receptor type 5(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50534982(CHEMBL4439458)
Affinity DataKi:  2.16E+4nMAssay Description:Time-dependent irreversible inhibition of N-terminal His-tagged STEP catalytic domain (unknown origin) expressed in Escherichia coli BL21 (DE3) cells...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141329(2-Benzenesulfonylamino-3-{4-[3-(1,4,5,6-tetrahydro...)
Affinity DataIC50:  0.110nMAssay Description:Binding affinity towards alpha V/beta3 receptor by solid-phase receptor binding assays (SPRA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141329(2-Benzenesulfonylamino-3-{4-[3-(1,4,5,6-tetrahydro...)
Affinity DataIC50:  0.120nMAssay Description:Binding affinity towards alpha V-beta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141324(2-Isopropoxycarbonylamino-3-{2-methoxy-4-[3-(1,4,5...)
Affinity DataIC50:  0.160nMAssay Description:Binding affinity towards alpha V/beta3 receptor by solid-phase receptor binding assays (SPRA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target72 kDa type IV collagenase(Homo sapiens (Human))
Fudan University

Curated by ChEMBL
LigandPNGBDBM50156468(CHEMBL3792916)
Affinity DataIC50:  0.190nMAssay Description:Inhibition of human recombinant MMP2 using Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg-NH2 as substrate preincubated for 60 mins followed by substrate addition b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141309(2-Benzenesulfonylamino-3-[4-(3-guanidino-benzoylam...)
Affinity DataIC50:  0.200nMAssay Description:Binding affinity towards alpha V/beta3 receptor by solid-phase receptor binding assays (SPRA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209479((beta1S)-3-bromo-5-chloro-b-[[[[3-[(5-fluoro-1,4,5...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209482((3S)-3-(5-chloro-2-hydroxy-3-methylphenyl)-3-(2-(3...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50185450(3-(benzo[d][1,3]dioxol-5-yl)-4-(1-methyl-5-(2-(5,6...)
Affinity DataIC50:  0.210nMAssay Description:Inhibition of alphavbeta3 integrin in 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141325(2-Benzenesulfonylamino-3-{4-[3-(4,5-dihydro-1H-imi...)
Affinity DataIC50:  0.270nMAssay Description:Binding affinity towards alpha V/beta3 receptor by solid-phase receptor binding assays (SPRA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209446((3S)-3-(3,5-dichloro-2-hydroxyphenyl)-3-(2-(3-(5-h...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209459((3R)-3-(2-(3-amino-5-(5-hydroxy-1,4,5,6-tetrahydro...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209471((3S)-3-(5-bromo-3-chloro-2-hydroxyphenyl)-3-(2-(3-...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141356(3-{3-Chloro-4-[3-(4,5-dihydro-1H-imidazol-2-ylamin...)
Affinity DataIC50:  0.310nMAssay Description:Binding affinity towards alpha V-beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141355(3-[4-(3-Guanidino-benzoylamino)-2-methoxy-phenyl]-...)
Affinity DataIC50:  0.320nMAssay Description:Binding affinity towards alpha V/beta3 receptor by solid-phase receptor binding assays (SPRA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50185464(3-(benzo[d][1,3]dioxol-5-yl)-4-(3-(2-(5,6,7,8-tetr...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of alphavbeta3 integrin in 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141324(2-Isopropoxycarbonylamino-3-{2-methoxy-4-[3-(1,4,5...)
Affinity DataIC50:  0.350nMAssay Description:Binding affinity towards alpha V-beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50141355(3-[4-(3-Guanidino-benzoylamino)-2-methoxy-phenyl]-...)
Affinity DataIC50:  0.380nMAssay Description:Binding affinity towards alpha V-beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209124((2,2-dimethyl-3-{4-[2-(5,6,7,8-tetrahydro-1,8-naph...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human intergrin alphavbeta3 receptor by solid phase receptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209124((2,2-dimethyl-3-{4-[2-(5,6,7,8-tetrahydro-1,8-naph...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human intergrin alphavbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209124((2,2-dimethyl-3-{4-[2-(5,6,7,8-tetrahydro-1,8-naph...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human intergrin alphavbeta3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209461((3S)-3-(3-bromo-5-chloro-2-hydroxyphenyl)-3-(2-(3-...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrin alpha-V/beta-3(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50209441((3S)-3-(3-bromo-5-chloro-2-hydroxyphenyl)-3-(2-(3-...)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of alphaVbeta3 integrin receptor expressed in human 293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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