Affinity DataKi: 0.0230nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0230nMAssay Description:Binding affinity of the compound towards human cloned B1 receptor was determined using [3H]-[des-Arg10-Leu9]-kallidin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0350nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
Affinity DataKi: 0.0600nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0640nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0650nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.0770nMAssay Description:Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.0800nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Binding affinity against rat Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity against human cloned Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Binding affinity to B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes.More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:The compound was evaluated for the inhibition of [125I]-Sar-AII binding to Angiotensin II receptor, type 1 from purified rat liver membranes.More data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 3.10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 4.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 5.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 5.60nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity towards human cloned Bradykinin receptor B2 expressed in CHO cells by [3H]bradykinin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: 9.16nMAssay Description:Binding affinity of the compound towards human cloned B2 receptor was determined using [3H]-BK as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Ability to bind to human cloned B2 receptor in competition binding experiments with [3H]- bradykininMore data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataKi: >10nMAssay Description:Ability to bind to human cloned B1 receptor in competition binding experiments with [3H][des-Arg10,Leu9]-Kallidin.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]des-Arg10-KD from human recombinant B1 receptor expressed in HEK293 cells by liquid scintillation counterMore data for this Ligand-Target Pair