Compile Data Set for Download or QSAR
maximum 50k data
Found 225 with Last Name = 'müller' and Initial = 'f'
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  0.390nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216040(3-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)quin...)
Affinity DataKi:  1.20nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219137(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216045(2-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-1,2...)
Affinity DataKi:  4.10nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50378584(STEPHOLIDINE)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219142(3-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dibe...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50378584(STEPHOLIDINE)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216046(2-(4-(4-phenyl-1-piperazinyl)butyl)-1,2-benzisothi...)
Affinity DataKi:  6.20nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219137(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  11.3nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50184429(16-methoxy-11-methyl-11-aza-tricyclo[12.4.0.03,8]o...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50010686((6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydr...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]spiperone from rat dopamine D4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219138(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  13.9nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216044(2-(4-(4-(3-a,a,a-trifluorotolyl)-1-piperazinyl)but...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(RAT)
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50010686((6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydr...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219138(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  17nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  17.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219142(3-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dibe...)
Affinity DataKi:  18.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219148(3-methoxy-8-methyl-5,6,7,8,9,10,11,16-octahydrodib...)
Affinity DataKi:  23.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50219140(12-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dib...)
Affinity DataKi:  25nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216044(2-(4-(4-(3-a,a,a-trifluorotolyl)-1-piperazinyl)but...)
Affinity DataKi:  26nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50184429(16-methoxy-11-methyl-11-aza-tricyclo[12.4.0.03,8]o...)
Affinity DataKi:  28.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219140(12-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dib...)
Affinity DataKi:  29.4nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50378584(STEPHOLIDINE)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216047(2-(4-(4-phenyl-1-piperazinyl)butyl)-1-isoindolinon...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50216052(2-(4-(4-(4-chlorophenyl)-1-piperazinyl)butyl)-1-is...)
Affinity DataKi:  33.6nMAssay Description:Displacement of [3H]SCH 23390 from human Dopamine D5 receptor expressed in HEK293More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216047(2-(4-(4-phenyl-1-piperazinyl)butyl)-1-isoindolinon...)
Affinity DataKi:  34nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50010686((6aR,12bS)-10,11-Dihydroxy-5,6,6a,7,8,12b-hexahydr...)
Affinity DataKi:  35.7nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216048(2-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-1-i...)
Affinity DataKi:  35.8nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216045(2-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-1,2...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50304398(5,8,13,13a-Tetrahydro-6H-isoquino[3,2-a]isoquinoli...)
Affinity DataKi:  41.1nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50184429(16-methoxy-11-methyl-11-aza-tricyclo[12.4.0.03,8]o...)
Affinity DataKi:  43.4nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216041(3-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)quin...)
Affinity DataKi:  46nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50180913(11-methyl-11-aza-tricyclo[12.4.0.0.3,8]octadeca-1(...)
Affinity DataKi:  47.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219148(3-methoxy-8-methyl-5,6,7,8,9,10,11,16-octahydrodib...)
Affinity DataKi:  53nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50184429(16-methoxy-11-methyl-11-aza-tricyclo[12.4.0.03,8]o...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50184429(16-methoxy-11-methyl-11-aza-tricyclo[12.4.0.03,8]o...)
Affinity DataKi:  54nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219140(12-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dib...)
Affinity DataKi:  55nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216048(2-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-1-i...)
Affinity DataKi:  60nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219137(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  60.1nMAssay Description:Displacement of [3H]spiperone from human dopamine D4.4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50219145(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  63nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216045(2-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)-1,2...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219145(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena

Curated by ChEMBL
LigandPNGBDBM50219145(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  70nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50216053(3-(4-(4-(3-a,a,a-trifluorotolyl)-1-piperazinyl)but...)
Affinity DataKi:  73nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50219137(7-methyl-6,7,8,9,10,15-hexahydro-5H-dibenzo[d,g]az...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50219149(2-methoxy-7-methyl-6,7,8,9,10,15-hexahydro-5H-dibe...)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena

Curated by ChEMBL
LigandPNGBDBM50216047(2-(4-(4-phenyl-1-piperazinyl)butyl)-1-isoindolinon...)
Affinity DataKi:  75.4nMAssay Description:Displacement of [3H]SCH 23390 from human Dopamine D5 receptor expressed in HEK293More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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