TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 0.390nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 3.20nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 5.90nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 9.80nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 11.3nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:Displacement of [3H]spiperone from rat dopamine D4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 13.9nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [3H]SCH23390 from rat dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 18.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 23.5nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 28.5nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 29.4nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]spiperone from rat dopamine D3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 33.6nMAssay Description:Displacement of [3H]SCH 23390 from human Dopamine D5 receptor expressed in HEK293More data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 35.7nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D1 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 35.8nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 41.1nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 43.4nMAssay Description:Displacement of [3H]spiperone from human dopamine D4 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 47.5nMAssay Description:Displacement of [3H]spiperone from human dopamine D3 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 54nMAssay Description:Displacement of [3H]SCH23390 from human dopamine D5 receptor expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 55nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Antagonist activity at human Dopamine receptor D2 isoform long expressed in HEK293 cells assessed as change in quinpirole-induced intracellular calci...More data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 60.1nMAssay Description:Displacement of [3H]spiperone from human dopamine D4.4 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 63nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 66nMAssay Description:Displacement of [3H]Spiperone from human Dopamine D3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Friedrich-Schiller-Universit£T Jena
Curated by ChEMBL
Affinity DataKi: 70nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 73nMAssay Description:Displacement of [3H]Spiperone from human Dopamine receptor D2 isoform long expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Displacement of [3H]spiperone from human dopamine D2L receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 75nMAssay Description:Displacement of [3H]SCH 23390 from human dopamine D5 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Friedrich-Schiller-UniversitäT Jena
Curated by ChEMBL
Affinity DataKi: 75.4nMAssay Description:Displacement of [3H]SCH 23390 from human Dopamine D5 receptor expressed in HEK293More data for this Ligand-Target Pair