Compile Data Set for Download or QSAR
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Found 211 with Last Name = 'müller' and Initial = 'w'
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151885(1-[4-(2,2-Diphenyl-ethylamino)-3-(morpholine-4-car...)
Affinity DataKi:  1nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151894(1-[4-(2,2-Diphenyl-ethylamino)-3-nitro-benzenesulf...)
Affinity DataKi:  10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151884(CHEMBL185551 | N,N-Bis-(3-dimethylamino-propyl)-3-...)
Affinity DataKi:  10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151891(CHEMBL273869 | {2-(2,2-Diphenyl-ethylamino)-5-[4-(...)
Affinity DataKi:  10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151886(CHEMBL181695 | {2-(2,2-Diphenyl-ethylamino)-5-[4-(...)
Affinity DataKi:  10nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151888(3-[3-Acetyl-4-(2,2-diphenyl-ethylamino)-benzenesul...)
Affinity DataKi:  130nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151889(CHEMBL180143 | N,N-Bis-(3-dimethylamino-propyl)-3-...)
Affinity DataKi:  140nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151890(CHEMBL181098 | N,N-Bis-(3-dimethylamino-propyl)-4-...)
Affinity DataKi:  230nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151893(4-(1-Benzyl-2-phenyl-ethylamino)-N,N-bis-(3-dimeth...)
Affinity DataKi:  250nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151892(3-[3-Chloro-4-(2,2-diphenyl-ethylamino)-benzenesul...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151887(4-(Benzhydryl-amino)-N,N-bis-(3-dimethylamino-prop...)
Affinity DataKi:  1.40E+3nMAssay Description:Binding affinity for Bradykinin receptor B2 expressed in COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB1 bradykinin receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50151887(4-(Benzhydryl-amino)-N,N-bis-(3-dimethylamino-prop...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity for Bradykinin receptor B1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  100nMAssay Description:Inhibition of aurora-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350423(CHEMBL466154)
Affinity DataIC50:  300nMAssay Description:Inhibition of recombinant PIM1 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  500nMAssay Description:Inhibition of aurora-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant Aurora-b assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  600nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  600nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  600nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  700nMAssay Description:Inhibition of SAK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  700nMAssay Description:Inhibition of SRC (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  800nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  800nMAssay Description:Inhibition of recombinant VEGF-R2 assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  800nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50446566(CHEMBL3109401)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant ALK (unknown origin) assessed as incorporation of [gamma-33P]-ATP into substrate by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetALK tyrosine kinase receptor(Homo sapiens (Human))
Heinrich Heine Universit£T

Curated by ChEMBL
LigandPNGBDBM50350424(CHEMBL454440)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of recombinant ALK assessed as 33Pi incorporation after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of MET (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428740(Bastadin 16 | CHEMBL2333164)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of aurora-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of COT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50150778(Bastadin-7 | Bastadins 7 | CHEMBL360190 | bastadin...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of CDK4/cyclin-D1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of INSR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of FLT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of CDK4/cyclin-D1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50150778(Bastadin-7 | Bastadins 7 | CHEMBL360190 | bastadin...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase kinase kinase 8(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of COT (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of VEGFR3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A1/Cyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of CDK2/cyclin-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428740(Bastadin 16 | CHEMBL2333164)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of aurora-B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428738(CHEMBL2333163 | Sesquibastadin 1)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of ARK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInsulin-like growth factor 1 receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50150778(Bastadin-7 | Bastadins 7 | CHEMBL360190 | bastadin...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of IGF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50241984(BASTADIN 6 | CHEMBL505907 | bastadin-6)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of aurora-A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of ARK5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiopoietin-1 receptor(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50150778(Bastadin-7 | Bastadins 7 | CHEMBL360190 | bastadin...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of TIE2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK4(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50150778(Bastadin-7 | Bastadins 7 | CHEMBL360190 | bastadin...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of SAK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Heinrich-Heine University

Curated by ChEMBL
LigandPNGBDBM50428737(BASTADIN 3)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of AKT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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