TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 0.00500nM ΔG°: -65.6kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 0.0620nM ΔG°: -59.2kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 0.0700nM ΔG°: -58.9kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 0.220nM ΔG°: -56.0kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 0.220nM ΔG°: -56.0kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 0.490nM ΔG°: -54.0kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Abbott Laboratories
Abbott Laboratories
Affinity DataKi: 2nM ΔG°: -50.5kJ/molepH: 4.7 T: 2°CAssay Description:HIV-1 protease activity was measured by a continuous fluorometric assay using the internally quenched fluorogenic substrate DABCYL-GABA-Ser-Gln-Tyr-P...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 30nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 45nM ΔG°: -41.5kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 57nM ΔG°: -40.9kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 79nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 150nM ΔG°: -38.6kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 220nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 240nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 260nM ΔG°: -37.2kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 270nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 310nM ΔG°: -36.8kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 350nM ΔG°: -36.5kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 350nM ΔG°: -36.5kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 370nM ΔG°: -36.3kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 470nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 490nM ΔG°: -35.7kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 610nM ΔG°: -35.1kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 610nM ΔG°: -35.1kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 660nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 830nM ΔG°: -34.4kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 1.56E+3nM ΔG°: -32.8kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+3nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 4.60E+3nMAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 6.67E+3nM ΔG°: -29.2kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 1.24E+4nM ΔG°: -27.7kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: 1.51E+4nM ΔG°: -27.2kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataKi: >4.00E+4nM ΔG°: >-24.8kJ/molepH: 7.5 T: 2°CAssay Description:A fluorogenic assay was used to measure influenza virus neuraminidase activity. The substrate, 4-methylumbelliferyl-N-acetylneuraminic acid, is cleav...More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of HCV 1b NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Inhibition of HCV 1a NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Inhibition of HCV 1b NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of HCV 1a NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 5.5nMAssay Description:Inhibition of HCV 1a NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of HCV 1b NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 6.70nMAssay Description:Inhibition of HCV 1b NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 8.70nMAssay Description:Inhibition of HCV 1a NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of HCV 1a NS5B RNA polymeraseMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of HCV 1a NS5B RNA polymeraseMore data for this Ligand-Target Pair