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Found 134 with Last Name = 'madison' and Initial = 'vs'
TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM50176988(8-Chloro-1-(2,4-dichloro-phenyl)-1,3a,4,5,6,10b-he...)
Affinity DataKi:  0.000350nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.98nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  2.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87019(1-(2,4-dichlorophenyl)-4-(hydroxymethyl)-N-(piperi...)
Affinity DataKi:  5.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM29094((+/-)-SLV319 | (S)-3-(4-chlorophenyl)-N-(4-chlorop...)
Affinity DataKi:  7.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP2/CNR2(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM50176988(8-Chloro-1-(2,4-dichloro-phenyl)-1,3a,4,5,6,10b-he...)
Affinity DataKi:  21nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87017(CAS_44450408 | NSC_44450408 | S-(R)-1-((2S,3R)-1-(...)
Affinity DataKi:  52.8nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM50080103(5,5-Bis-(4-bromo-phenyl)-3-(2-morpholin-4-yl-ethyl...)
Affinity DataKi:  70.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444918(CHEMBL3099753)
Affinity DataKi: <100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87015(1-(bis(4-chlorophenyl)methyl)-3-((3,5-difluorophen...)
Affinity DataKi:  100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444921(CHEMBL3099750)
Affinity DataKi:  100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444933(CHEMBL3099763)
Affinity DataKi: <100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444932(CHEMBL3099764)
Affinity DataKi: <100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444934(CHEMBL3099762)
Affinity DataKi: <100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444935(CHEMBL3099761)
Affinity DataKi: <100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444919(CHEMBL3099752)
Affinity DataKi:  100nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171301((S)-(2-{3-[((9S,12S)-12-Cyclohexyl-11,14-dioxo-2-o...)
Affinity DataKi:  110nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444941(CHEMBL3099755)
Affinity DataKi:  140nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetGTP-binding nuclear protein GSP1/CNR1(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87014(4-(6-methoxy-2-(4-methoxyphenyl)benzofuran-3-carbo...)
Affinity DataKi:  141nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444920(CHEMBL3099751)
Affinity DataKi:  160nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171302((S)-(2-{3-[((9S,12S)-12-Cyclohexyl-11,14-dioxo-2-o...)
Affinity DataKi:  160nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87013((3R,4S)-3-(benzofuran-2-ylmethyl)-4-(4-methoxyphen...)
Affinity DataKi:  194nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444938(CHEMBL3099758)
Affinity DataKi:  200nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87020((3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin...)
Affinity DataKi:  244nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87017(CAS_44450408 | NSC_44450408 | S-(R)-1-((2S,3R)-1-(...)
Affinity DataKi:  282nMMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444922(CHEMBL3099749)
Affinity DataKi:  300nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171302((S)-(2-{3-[((9S,12S)-12-Cyclohexyl-11,14-dioxo-2-o...)
Affinity DataKi:  300nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-chlorophenylbutyric acid ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV proteas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171305((S)-(2-{3-[((9S,12S)-12-Cyclohexyl-11,14-dioxo-2-o...)
Affinity DataKi:  300nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87018((3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3...)
Affinity DataKi:  301nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87016(4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)...)
Affinity DataKi:  452nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  560nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444940(CHEMBL3099756)
Affinity DataKi:  700nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50370596(CHEMBL1169404)
Affinity DataKi:  800nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444939(CHEMBL3099757)
Affinity DataKi:  900nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444942(CHEMBL3099754)
Affinity DataKi:  900nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP2/CNR2(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87020((3R,4S)-4-(4-methoxyphenyl)-1-phenyl-3-(3-(pyridin...)
Affinity DataKi:  1.09E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87016(4-(4-methoxyphenyl)-1-phenyl-3-(2-(phenylsulfonyl)...)
Affinity DataKi:  1.24E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87018((3S,4R)-1-(4-fluorophenyl)-3-(3-(4-fluorophenyl)-3...)
Affinity DataKi:  1.82E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP2/CNR2(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87019(1-(2,4-dichlorophenyl)-4-(hydroxymethyl)-N-(piperi...)
Affinity DataKi:  2.31E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444923(CHEMBL3099748)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444928(CHEMBL3099743)
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444936(CHEMBL3099760)
Affinity DataKi:  2.80E+3nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171301((S)-(2-{3-[((9S,12S)-12-Cyclohexyl-11,14-dioxo-2-o...)
Affinity DataKi:  2.90E+3nMAssay Description:Binding constant towards Human neutrophil elastase HNE proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171304((S)-(2-{(S)-3-[((9S,12S,15S)-15-tert-Butoxycarbony...)
Affinity DataKi:  7.80E+3nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP2/CNR2(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM29094((+/-)-SLV319 | (S)-3-(4-chlorophenyl)-N-(4-chlorop...)
Affinity DataKi:  7.94E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGTP-binding nuclear protein GSP2/CNR2(Saccharomyces cerevisiae)
Cns Biological Research

Curated by PDSP Ki Database
LigandPNGBDBM87014(4-(6-methoxy-2-(4-methoxyphenyl)benzofuran-3-carbo...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444937(CHEMBL3099759)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50444924(CHEMBL3099747)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of B-Alexa-Fluor647 from CDK2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Hepatitis C virus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50171303(CHEMBL370096 | {3-[((9S,12S,15S)-15-tert-Butoxycar...)
Affinity DataKi:  1.20E+4nMAssay Description:Ability to inhibit the hydrolysis of chromogenic 4-phenylazophenyl ester from the peptide fragment Ac- DTEDVVP(Nva)-O-4-PAP in a HCV protease continu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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