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Found 101 with Last Name = 'maeda' and Initial = 'j'
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.0430nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185958(CHEMBL205971 | N-(2-methoxybenzyl)-N-(4-chloro-2-p...)
Affinity DataKi:  0.0700nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185958(CHEMBL205971 | N-(2-methoxybenzyl)-N-(4-chloro-2-p...)
Affinity DataKi:  0.0740nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122294(CHEMBL292092 | N-(5-fluoro-2-phenoxyphenyl)-N-(2-(...)
Affinity DataKi:  0.0780nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185959(CHEMBL381602 | N-(2-ethoxybenzyl)-N-(4-chloro-2-ph...)
Affinity DataKi:  0.0980nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185959(CHEMBL381602 | N-(2-ethoxybenzyl)-N-(4-chloro-2-ph...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.100nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.160nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [11C]DAA1106 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122295(CHEMBL63065 | N-(2-Fluoromethoxy-5-methoxy-benzyl)...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50122293(CHEMBL401000 | CHEMBL63064 | N-(2,5-Dimethoxy-benz...)
Affinity DataKi:  0.188nMAssay Description:In vitro binding affinity for PBR (peripheral benzodiazepine receptor) in monkey brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185957(CHEMBL205767 | N-(2-isopropoxybenzyl)-N-(4-chloro-...)
Affinity DataKi:  0.190nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312840(CHEMBL1076680 | US9139546, 16 | [11C](3',5'-dichlo...)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to rat brain CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50163592((3,4-Dihydro-2H-1-oxa-9-aza-anthracen-6-yl)-(4-met...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329410(CHEMBL1270323 | N-(2-(4-(benzo[d]isoxazol-3-yl)pip...)
Affinity DataKi:  0.340nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50301822(5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  0.540nMAssay Description:Displacement of [11C](R)-PK1119 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50185957(CHEMBL205767 | N-(2-isopropoxybenzyl)-N-(4-chloro-...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [11C]DAA1106 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  0.820nMAssay Description:Displacement of [11C]DAA1106 from Sprague-Dawley rat brain PBRMore data for this Ligand-Target Pair
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM22032(1-(2-chlorophenyl)-N-methyl-N-(1-methylpropyl)isoq...)
Affinity DataKi:  0.830nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333368(CHEMBL1645348 | [11C]-cis-(3-ethyl-2-methylquinoli...)
Affinity DataKi:  0.870nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329412(CHEMBL1270423 | N-[2-[4-(3-Cyanopyridin-2-yl)piper...)
Affinity DataKi:  0.930nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329407(CHEMBL1270121 | N-[2-[4-(3-Cyanopyridin-2-yl)piper...)
Affinity DataKi:  1.52nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329408(CHEMBL1270227 | N-[2-[4-(4-Chlorophenyl)piperazin-...)
Affinity DataKi:  1.76nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329405(CHEMBL1270013 | N-(2-(4-(benzo[d]isoxazol-3-yl)pip...)
Affinity DataKi:  1.93nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312841(CHEMBL1081609 | US9139546, 30 | [11C](3',5'-dichlo...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity to rat brain CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329409(CHEMBL1270322 | N-[2-[4-(4-Methylphenyl)piperazin-...)
Affinity DataKi:  2.64nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329413(CHEMBL1270516 | N-[2-[4-(5-Chloropyridin-2-yl)pipe...)
Affinity DataKi:  2.92nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50273942(4-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190677((R)-3'-(3-bromobenzo[b]thiophen-5-yl)spiro[1-azabi...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190696((2S)-3'-(5-bromothien-2-yl)-2'H-spiro[4-azabicyclo...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190686((R)-3'-(2,3-dimethylbenzo[b]thiophen-5-yl)spiro[1-...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312838(CHEMBL1081623 | SCH-225336 | [11C]N-(1-(4-(4-metho...)
Affinity DataKi:  4.5nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50144889(CHEMBL72521 | N-(5-Fluoro-2-phenoxy-phenyl)-N-(2-i...)
Affinity DataKi:  4.80nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50333371(CHEMBL1645351 | CHEMBL1771388 | [11C]-6-N-cyclohex...)
Affinity DataKi:  4.80nMAssay Description:Binding affinity to mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50068366(CHEMBL93403 | N-{2-[4-(4-Chloro-phenyl)-piperazin-...)
Affinity DataKi:  4.97nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50122028(3-Methoxy-N-[2-(4-p-tolyl-piperazin-1-yl)-ethyl]-b...)
Affinity DataKi:  9.21nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312837(CHEMBL1081610 | [11C]8-butoxy-N-cyclohexyl-7-metho...)
Affinity DataKi:  9.60nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50122044(CHEMBL345111 | N-{2-[4-(5-Chloro-pyridin-2-yl)-pip...)
Affinity DataKi:  11.3nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400331(CHEMBL2181520)
Affinity DataKi:  13.6nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranslocator protein(Rattus norvegicus (rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50144887(CHEMBL443526 | Toluene-4-sulfonic acid 2-(2-{[acet...)
Affinity DataKi:  18.1nMAssay Description:In vitro inhibition of [11C]2 binding to Peripheral benzodiazepine receptor (PBR) in rat brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400332(CHEMBL2181521)
Affinity DataKi:  22.2nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50400330(CHEMBL2181519)
Affinity DataKi:  27.3nMAssay Description:Displacement of [18F]FITM from mGlu1 receptor in rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329411(CHEMBL1270422 | N-[2-[4-(4-Cyanophenyl)piperazin-1...)
Affinity DataKi:  32.7nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312839(CHEMBL1081622 | [18F]8-butoxy-N-cyclohexyl-7-(2-fl...)
Affinity DataKi:  36nMAssay Description:Binding affinity to human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
Universita` Degli Studi Di Bari A Moro

Curated by ChEMBL
LigandPNGBDBM50329406(CHEMBL1270120 | N-[2-[4-(4-Cyanophenyl)piperazin-1...)
Affinity DataKi:  64.0nMAssay Description:Displacement of [3H]MSP from rat dopamine D4 receptor expressed in HEK293 cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Mitsubishi Pharma

Curated by ChEMBL
LigandPNGBDBM50190687((R)-3'-(indan-5-yl)spiro[-1-azabicyclo[2.2.2]octan...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]alpha-BTX from alpha-7 nAChR in rat hippocampus membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312841(CHEMBL1081609 | US9139546, 30 | [11C](3',5'-dichlo...)
Affinity DataKi:  503nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50312840(CHEMBL1076680 | US9139546, 16 | [11C](3',5'-dichlo...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSignal transducer and activator of transcription 6(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50304425(2-(4-morpholinophenylamino)-4-(2,3,6-trifluorobenz...)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of STAT6 in IL4-stimulated human FW4 reporter cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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