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Found 239 with Last Name = 'maeng' and Initial = 'jh'
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM93624(5-methyl-2-[(5-methyl-1H-imidazol-4-yl)methyl]-3,4...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329746(CHEMBL1271731 | endo-2-((3S,5S)-3,5-dimethylmorpho...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329748(CHEMBL1271791 | endo-2-((3S,5S)-3-ethyl-5-methylmo...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329745(CHEMBL1271730 | endo-2-((S)-3-tert-butylmorpholino...)
Affinity DataKi:  2nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329724(CHEMBL1271960 | endo-2-((2S,6S)-2,6-dimethylpipera...)
Affinity DataKi:  2.40nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  3.40nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329744(CHEMBL1271678 | endo-2-((S)-3-isobutylmorpholino)-...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329742(CHEMBL1271629 | endo-N-((1R,5R)-9-methyl-9-azabicy...)
Affinity DataKi:  3.90nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329741(CHEMBL1271628 | endo-2-((S)-3-ethylmorpholino)-N-(...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329730((S)-2-amino-6-chloro-N-(quinuclidin-3-yl)benzo[d]o...)
Affinity DataKi:  4.70nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329743(CHEMBL1271677 | endo-2-((S)-3-isopropylmorpholino)...)
Affinity DataKi:  5nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329747(2-((3S,5S)-3,5-dimethylmorpholino)-N-((S)-quinucli...)
Affinity DataKi:  6.80nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329728(CHEMBL1272073 | endo-2-cyclopropyl-N-((1R,5R)-9-me...)
Affinity DataKi:  8.30nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329754((S)-2-(diethylamino)-N-(quinuclidin-3-yl)benzo[d]o...)
Affinity DataKi:  12.4nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329739(CHEMBL1271570 | endo-N-(8-methyl-8-azabicyclo[3.2....)
Affinity DataKi:  12.9nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329729((S)-2-amino-N-(quinuclidin-3-yl)benzo[d]oxazole-4-...)
Affinity DataKi:  13.8nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329726(CHEMBL1272017 | endo-2-(2-methoxyphenyl)-N-((1R,5R...)
Affinity DataKi:  14.9nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329731(CHEMBL1272174 | endo-N-((1R,5R)-9-methyl-9-azabicy...)
Affinity DataKi:  15.1nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329732(CHEMBL1272175 | endo-2-(4-fluorophenyl)-N-((1R,5R)...)
Affinity DataKi:  16.3nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329751(CHEMBL1271904 | endo-N-((1R,5R)-9-methyl-9-azabicy...)
Affinity DataKi:  16.5nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329733(CHEMBL1272230 | endo-2-(4-chlorophenyl)-N-((1R,5R)...)
Affinity DataKi:  18nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329756((S)-2-(dimethylamino)-N-(quinuclidin-3-yl)benzo[d]...)
Affinity DataKi:  18.2nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329734(CHEMBL1272231 | endo-2-(4-methoxyphenyl)-N-((1R,5R...)
Affinity DataKi:  18.8nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329727((S)-2-cyclopropyl-N-(quinuclidin-3-yl)benzo[d]oxaz...)
Affinity DataKi:  32.7nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329749(CHEMBL1271848 | endo-2-((2R,6S)-2,6-dimethylmorpho...)
Affinity DataKi:  35.3nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329758((S)-2-(methylamino)-N-(quinuclidin-3-yl)benzo[d]ox...)
Affinity DataKi:  36.4nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329757((S)-2-(ethylamino)-N-(quinuclidin-3-yl)benzo[d]oxa...)
Affinity DataKi:  36.4nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329752(CHEMBL1271905 | endo-2-((2S,6R)-2,6-dimethylpipera...)
Affinity DataKi:  37.3nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329722(CHEMBL1271519 | endo-N-((1R,5R)-9-methyl-9-azabicy...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329735(CHEMBL1272283 | endo-N-((1R,5R)-9-methyl-9-azabicy...)
Affinity DataKi:  40.4nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329725((S)-2-(2-methoxyphenyl)-N-(quinuclidin-8-yl)benzo[...)
Affinity DataKi:  47.3nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329738(CHEMBL1271466 | endo-2-(4-methoxyphenyl)-N-((1R,5R...)
Affinity DataKi:  58.5nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329753(CHEMBL1271959 | endo-2-((2R,6R)-2,6-dimethylpipera...)
Affinity DataKi:  59.4nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329755(2-(1-(methylamino)ethyl)-N-((S)-quinuclidin-3-yl)b...)
Affinity DataKi:  66.5nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329750(CHEMBL1271849 | endo-N-((1R,5R)-9-methyl-9-azabicy...)
Affinity DataKi:  72.2nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329737(CHEMBL1271465 | endo-2-(4-chlorophenyl)-N-((1R,5R)...)
Affinity DataKi:  73.8nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329740(CHEMBL1271571 | N-((1R,5R)-9-methyl-9-azabicyclo[3...)
Affinity DataKi:  92.6nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329736(CHEMBL1272284 | endo-2-(4-fluorophenyl)-N-((1R,5R)...)
Affinity DataKi:  94.9nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50329723((S)-2-morpholino-N-(quinuclidin-3-yl)benzo[d]oxazo...)
Affinity DataKi:  165nMAssay Description:Binding affinity to human HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533742(CHEMBL4593786)
Affinity DataIC50:  0.671nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533732(CHEMBL4526580)
Affinity DataIC50:  0.726nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533748(CHEMBL4468117)
Affinity DataIC50:  0.733nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM20880((2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)me...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human SGLT2 expressed in CHOK1 cells assessed as inhibition of [14C]-AMG uptake after 3 hrs by microbeta scintillation counting analysi...More data for this Ligand-Target Pair
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533727(CHEMBL4456392)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533730(CHEMBL4582587)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533749(CHEMBL4516089)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533723(CHEMBL4572086)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533725(CHEMBL4579165)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533736(CHEMBL4462009)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium- and chloride-dependent glycine transporter 1(Homo sapiens (Human))
Amri

Curated by ChEMBL
LigandPNGBDBM50533733(CHEMBL4532784)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of glycine transporter-1B in human JAR cells assessed as reduction in [14C]glycine uptake preincubated for 10 mins followed by [14C]glycin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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