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Found 195 with Last Name = 'mahale' and Initial = 's'
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188069(12-oxo-10,12-dihydro-10-aza-4b-azonia-indeno[2,1-b...)
Affinity DataIC50:  410nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM59087(CHEMBL258765 | Fasca-plysi | Fascaplysin)
Affinity DataIC50:  410nMAssay Description:Binding affinity to human CDK4/cyclinD1 using GST-pRB152 as substrate by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM59087(CHEMBL258765 | Fasca-plysi | Fascaplysin)
Affinity DataIC50:  550nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM59087(CHEMBL258765 | Fasca-plysi | Fascaplysin)
Affinity DataIC50:  550nMAssay Description:Inhibition of human CDK4/ Cyclin D1 catalytic subunit expressed in Sf9 insect cells assessed as GST-RB152 fusion protein phosphorylation-associated d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50188071(CHEMBL213805 | biphenyl-4-carboxylic acid [2-(1H-i...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188071(CHEMBL213805 | biphenyl-4-carboxylic acid [2-(1H-i...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188071(CHEMBL213805 | biphenyl-4-carboxylic acid [2-(1H-i...)
Affinity DataIC50:  6.20E+3nMAssay Description:Binding affinity to human CDK4/cyclinD1 using GST-pRB152 as substrate by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273105((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-me...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272870(CHEMBL498710 | N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273041((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272800(CHEMBL498521 | N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273074((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-fl...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272837(CHEMBL496481 | N-(2-(1H-Indol-3-yl)ethyl)-4'-fluor...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272919(CHEMBL456121 | N-(2-(1H-Indol-3-yl)ethyl)-3'-methy...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272836(CHEMBL521733 | N-(2-(1H-Indol-3-yl)ethyl)biphenyl-...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273076((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-fl...)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272838(CHEMBL496482 | N-(2-(1H-Indol-3-yl)ethyl)-4'-methy...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273039((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-fl...)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272997((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-fl...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272918(CHEMBL456964 | N-(2-(1H-Indol-3-yl)ethyl)-3'-fluor...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272798(CHEMBL498520 | N-(2-(1H-Indol-3-yl)ethyl)-4'-fluor...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273075((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-fl...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273109((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-me...)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272995((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-fl...)
Affinity DataIC50:  2.30E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272799(CHEMBL525921 | N-(2-(1H-Indol-3-yl)ethyl)-N,4'-dim...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273040((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-me...)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272999((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(4'-fl...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273106((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273141(CHEMBL457179 | N-(2-(1H-Indol-3-yl)ethyl)-N-methyl...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272917(CHEMBL456760 | N-(2-(1H-Indol-3-yl)ethyl)-2'-metho...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272998((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273038((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-fl...)
Affinity DataIC50:  2.70E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273108((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273142(CHEMBL515051 | N-(2-(1H-Indol-3-yl)ethyl)-3-(pyrid...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273107((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2'-me...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273072((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-me...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272996((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(3'-fl...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272835(CHEMBL498705 | N-(2-(1H-Indol-3-yl)ethyl)-4'-pheny...)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273144((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2-(py...)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50297259(1,2-Bis-(indol-1-yl)-ethane | CHEMBL549792)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human CDK4/ Cyclin D1 catalytic subunit expressed in Sf9 insect cells assessed as GST-RB152 fusion protein phosphorylation-associated d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188075(CHEMBL378617 | N-(2-(1H-indol-3-yl)ethyl)-4-bromo-...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188066(CHEMBL213302 | N-(2-(1H-indol-3-yl)ethyl)-4-chloro...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of Cdk4/Cyclin D1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
De Montfort University

Curated by ChEMBL
LigandPNGBDBM50188066(CHEMBL213302 | N-(2-(1H-indol-3-yl)ethyl)-4-chloro...)
Affinity DataIC50:  3.80E+4nMAssay Description:Binding affinity to human CDK4/cyclinD1 using GST-pRB152 as substrate by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50297260(1,3-Bis-(indol-1-yl)-propane | CHEMBL557456)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human CDK4/ Cyclin D1 catalytic subunit expressed in Sf9 insect cells assessed as GST-RB152 fusion protein phosphorylation-associated d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50297274(1-(5-Methyl-2,3-dihydro-indol-1-yl)-2-(5-methyl-1H...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human CDK4/ Cyclin D1 catalytic subunit expressed in Sf9 insect cells assessed as GST-RB152 fusion protein phosphorylation-associated d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50297282(5-Chloro-3-[2-(5-chloro-3a,7a-dihydro-indol-1-yl)-...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human CDK4/ Cyclin D1 catalytic subunit expressed in Sf9 insect cells assessed as GST-RB152 fusion protein phosphorylation-associated d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272874(CHEMBL525530 | N-(2-(1H-Indol-3-yl)ethyl)-4'-tert-...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50272873(CHEMBL497454 | N-(2-(1H-Indol-3-yl)ethyl)-4'-fluor...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50273143((3,4-Dihydro-1H-pyrido[3,4-b]indol-2(9H)-yl)(2-(py...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of human CDK4/GST-cyclin D1 expressed in Sf9 cells assessed as retinoblastoma GST-RB152 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4(Homo sapiens (Human))
University Of Leicester

Curated by ChEMBL
LigandPNGBDBM50297268(1-(2,3-Dihydro-indol-1-yl)-2-(5-methyl-1H-indol-3-...)
Affinity DataIC50:  4.15E+4nMAssay Description:Inhibition of human CDK4/ Cyclin D1 catalytic subunit expressed in Sf9 insect cells assessed as GST-RB152 fusion protein phosphorylation-associated d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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