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Found 23 with Last Name = 'maitre' and Initial = 'm'
TargetGamma-hydroxybutyrate receptor(RAT)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50023573(4-Cyclohexyl-4-hydroxy-but-2-enoic acid | CHEMBL17...)
Affinity DataIC50:  3.30nMAssay Description:Binding affinity towards [3H]-GHB binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50023572(CHEMBL354804 | Sodium; 4-hydroxy-but-2-enoate)
Affinity DataIC50:  3.5nMAssay Description:Binding affinity towards [3H]-GHB binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50023574(4-Hydroxy-pent-2-enoic acid | CHEMBL171595)
Affinity DataIC50:  11nMAssay Description:Binding affinity towards [3H]-GHB binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-hydroxybutyrate receptor(RAT)
Centre De Neurochimie Du Cnrs

Curated by ChEMBL
LigandPNGBDBM50023575(4-hydroxy-butyric acid | 4-hydroxybutanoic acid | ...)
Affinity DataIC50:  6.60E+3nMAssay Description:Binding affinity towards [3H]-GHB binding siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084977(3,5,7-Trihydroxy-2-[3-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataKd:  250nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084978(3,5,7-trihydroxy-2-(4-methoxyphenyl)-4H-chromen-4-...)
Affinity DataKd:  4.50E+3nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084981(8-((E)-3,7-Dimethyl-octa-2,6-dienyl)-3,5,7-trihydr...)
Affinity DataKd:  120nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50218276(Silibinin | Silymarin)
Affinity DataKd:  6.80E+3nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50049400((+/-) taxifolin | (+/-)-Dihydroquercetin | (+/-)-t...)
Affinity DataKd:  3.74E+4nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50013111(1-((2R,5S)-5-(hydroxymethyl)-2,5-dihydrofuran-2-yl...)
Affinity DataEC50:  50nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044905((10,13-Dimethyl-17-octyl-2,3,4,7,8,9,10,11,12,13,1...)
Affinity DataEC50:  20nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044910(CHEMBL352398 | Phosphoric acid bis-[5-(5-methyl-2,...)
Affinity DataEC50:  50nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataEC50:  10nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044911(CHEMBL170331 | Heptadeca-9,12,15-trienoic acid 5-(...)
Affinity DataEC50:  40nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044906(CHEMBL353179 | Phosphoric acid 8-(10,13-dimethyl-3...)
Affinity DataEC50:  50nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044913(CHEMBL440551 | Heptadeca-9,12-dienoic acid 5-(5-me...)
Affinity DataEC50:  20nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044908(CHEMBL170006 | Phosphoric acid hexadecyl ester 5-(...)
Affinity DataEC50:  200nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Ura Cnrs 1309

Curated by ChEMBL
LigandPNGBDBM50044907(CHEMBL166614 | Hexadecanoic acid 5-(5-methyl-2,4-d...)
Affinity DataEC50:  80nMAssay Description:Effective concentration that reduces HIV-induced cytopathic effect by 50% was determined by reverse transcriptase (RT) assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084976(3,5,7-Trihydroxy-2-[3-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataKd:  370nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM23419((2S)-5,7-dihydroxy-2-(4-hydroxyphenyl)-3,4-dihydro...)
Affinity DataKd:  2.85E+4nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084975(6-((E)-3,7-Dimethyl-octa-2,6-dienyl)-3,5,7-trihydr...)
Affinity DataKd:  180nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM18627((10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]...)
Affinity DataKd:  2.00E+4nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Mus musculus (Mouse))
Universit£

Curated by ChEMBL
LigandPNGBDBM50084979(3,5,7-Trihydroxy-2-[3-(4-hydroxy-3-methoxy-phenyl)...)
Affinity DataKd:  2.20E+3nMAssay Description:Compound was tested for the binding affinity towards recombinant NBD2 C-terminal cytotoxic nucleotide-binding domain of mouse P-GlycoproteinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed