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Found 38 with Last Name = 'marasco' and Initial = 'd'
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)
Affinity DataKi:  0.251nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)
Affinity DataKi:  0.398nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)
Affinity DataKi:  0.724nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)
Affinity DataKi:  0.776nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)
Affinity DataKi:  0.794nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048700(CHEMBL3315147)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)
Affinity DataKi:  1.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)
Affinity DataKi:  1.70nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048703(CHEMBL3315150)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048692(CHEMBL3315140)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048702(CHEMBL3315149)
Affinity DataKi:  2.20nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50411333(URANTIDE)
Affinity DataKi:  5nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048690(CHEMBL3315143)
Affinity DataKi:  6.5nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048704(CHEMBL3315151)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048698(CHEMBL3315145)
Affinity DataKi:  13nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(Homo sapiens (Human))
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048706(CHEMBL3315153)
Affinity DataKi:  17nMAssay Description:Displacement of [125I]urotensin-2 from human recombinant UT receptor expressed in CHO-K1 cells by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Indiana University School Of Medicine

LigandPNGBDBM119124((E)-2-[(4,5-Dimethoxy-2-methyl-3,6-dioxocyclohexa-...)
Affinity DataIC50:  8.50E+3nMpH: 7.5Assay Description:E3330 or E3330-amide was preincubated with 2 μL of APE1 (reduced with 1.0 mM DTT for 10 min and then diluted to a concentration of 0.06 mM with ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA-(apurinic or apyrimidinic site) endonuclease(Homo sapiens (Human))
Indiana University School Of Medicine

LigandPNGBDBM50303955((E)-3-(5,6-Dimethoxy-3-methyl-14-dioxocyclohexa-25...)
Affinity DataIC50:  2.00E+4nMpH: 7.5Assay Description:E3330 or E3330-amide was preincubated with 2 μL of APE1 (reduced with 1.0 mM DTT for 10 min and then diluted to a concentration of 0.06 mM with ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50578551(CHEMBL4851880)
Affinity DataKd:  3.50E+4nMAssay Description:Binding affinity to N-terminal His-tagged human JAK2 catalytic domain (826 to 1132 residues) expressed in baculovirus-infected Sf21 cells by Microsca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048690(CHEMBL3315143)
Affinity DataEC50:  18nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50320463(CHEMBL218994 | D[CFWKYC]V | H-Asp-Cys-Phe-Trp-Lys-...)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048691(CHEMBL3315139)
Affinity DataEC50:  0.398nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048692(CHEMBL3315140)
Affinity DataEC50:  0.724nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048695(CHEMBL3315141)
Affinity DataEC50:  3.80nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048696(CHEMBL3315142)
Affinity DataEC50:  5nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048698(CHEMBL3315145)
Affinity DataEC50:  34nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048697(CHEMBL3315144)
Affinity DataEC50:  0.0195nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048699(CHEMBL3315146)
Affinity DataEC50:  0.813nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048700(CHEMBL3315147)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048701(CHEMBL3315148)
Affinity DataEC50:  0.0126nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048702(CHEMBL3315149)
Affinity DataEC50:  13nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048703(CHEMBL3315150)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50048705(CHEMBL3315152)
Affinity DataEC50:  0.631nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50540551(CHEMBL4641893)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to human N-terminal His-tagged JAK2 catalytic domain (826 to 1132 end residues) at 25 degree C by microscale thermophoresis assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
University Of Naples "Federico Ii

Curated by ChEMBL
LigandPNGBDBM50578550(CHEMBL4857393)
Affinity DataKd:  4.40E+4nMAssay Description:Binding affinity to N-terminal His-tagged human JAK2 catalytic domain (826 to 1132 residues) expressed in baculovirus-infected Sf21 cells by Microsca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrotensin-2 receptor(RAT)
University Of Naples&Quot;Federico Ii&Quot

Curated by ChEMBL
LigandPNGBDBM50413784(UROTENSIN-II)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at UT receptor in rat aorta assessed as contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed