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Found 104 with Last Name = 'marks' and Initial = 'js'
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291640(CHEMBL274146 | Dipeptide Ligand)
Affinity DataIC50:  240nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287070((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[(R)-3-...)
Affinity DataIC50:  350nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060738(2-[2-(4-Carboxy-2-{4-carboxy-2-[(R)-3-carboxy-2-(4...)
Affinity DataIC50:  400nMAssay Description:Inhibition of [125I]-phosphopeptide binding to Src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  500nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to SRC SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  500nMAssay Description:Inhibition of [125I]-phosphopeptide binding to Src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50450413(CHEMBL328907)
Affinity DataIC50:  500nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060736((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  800nMAssay Description:Inhibition of [125I]-phosphopeptide binding to Src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289749(CHEMBL414123 | Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Il...)
Affinity DataIC50:  800nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to SRC SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289749(CHEMBL414123 | Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Il...)
Affinity DataIC50:  800nMAssay Description:Inhibition of [35S]-labeled SH2-GST Abl binding to the phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289743((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  800nMAssay Description:Inhibition of [35S]-labeled SH2-GST Abl binding to the phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289748((S)-2-{(2S,3S)-2-[(S)-2-((S)-2-{(S)-2-Acetylamino-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Abl binding to the phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289748((S)-2-{(2S,3S)-2-[(S)-2-((S)-2-{(S)-2-Acetylamino-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to ABL SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289747((S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Src binding to phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50450413(CHEMBL328907)
Affinity DataIC50:  1.35E+3nMAssay Description:Inhibition of src SH2 domain binding to PDGF receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287069((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[2-(2-h...)
Affinity DataIC50:  1.40E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289747((S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Abl binding to the phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Src binding to phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289746(CHEMBL298813 | {[4-((S)-2-Acetylamino-2-{(S)-1-[(3...)
Affinity DataIC50:  1.60E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to ABL SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289750((S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-...)
Affinity DataIC50:  1.70E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to ABL SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289743((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060734((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of [125I]-phosphopeptide binding to Src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289752(CHEMBL413629 | Glu-Pro-Gln-F2Pmp-Glu-Glu-Ile-Pro-I...)
Affinity DataIC50:  1.80E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to SRC SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289742((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  1.80E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to ABL SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291638((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060734((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287075((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[2-(3-h...)
Affinity DataIC50:  2.10E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287075((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[2-(3-h...)
Affinity DataIC50:  2.10E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289750((S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-...)
Affinity DataIC50:  2.10E+3nMAssay Description:Functional antagonism against ETA receptor in rat aortic rings expressed as pA2 valueMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291647(4-[2-Acetylamino-3-(4-phosphonooxy-phenyl)-propion...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50060735(2-[2-(2-{2-[(S)-2-Acetylamino-3-(4-phosphonooxy-ph...)
Affinity DataIC50:  2.80E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289749(CHEMBL414123 | Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Il...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Abl binding to the phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291651(4-[2-Acetylamino-3-(4-phosphonooxy-phenyl)-propion...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289750((S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-...)
Affinity DataIC50:  3.40E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to SRC SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287076((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[3-(4-p...)
Affinity DataIC50:  3.40E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291645(4-[2-Acetylamino-3-(4-phosphonooxy-phenyl)-propion...)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291650(CHEMBL13424 | Dipeptide Ligand)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287074(4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)-pro...)
Affinity DataIC50:  4.00E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289743((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  4.00E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to ABL SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289746(CHEMBL298813 | {[4-((S)-2-Acetylamino-2-{(S)-1-[(3...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Abl binding to the phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291641(4-[{2-[2-Acetylamino-3-(4-phosphonooxy-phenyl)-pro...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50118657(Ac-pYEEIE | CHEMBL2092742)
Affinity DataIC50:  4.50E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50118657(Ac-pYEEIE | CHEMBL2092742)
Affinity DataIC50:  4.50E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287077((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[3-(2,6...)
Affinity DataIC50:  4.50E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291642(4-[2-Acetylamino-3-(4-phosphonooxy-phenyl)-propion...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50291653(4-[2-Acetylamino-3-(4-phosphonooxy-phenyl)-propion...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of [125I]-labeled phosphopeptide binding to a Src protein tryrosine kinase SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289742((S)-4-[(S)-2-Acetylamino-3-(4-phosphonooxy-phenyl)...)
Affinity DataIC50:  4.90E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to ABL SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289747((S)-4-{(S)-2-Acetylamino-3-[4-(difluoro-phosphono-...)
Affinity DataIC50:  4.90E+3nMAssay Description:Radioligand displacement assay for the binding of [125I]-Glu-Pro-Gln-pTyr-Glu-Glu-Ile-Pro-Ile-Tyr-Leu to SRC SH2 domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287078((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[(Z)-2-...)
Affinity DataIC50:  5.00E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289748((S)-2-{(2S,3S)-2-[(S)-2-((S)-2-{(S)-2-Acetylamino-...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of [35S]-labeled SH2-GST Src binding to phospho-PDGF receptor intracellular domainMore data for this Ligand-Target Pair
In DepthDetails Article
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287082((S)-2-[(2S,3S)-2-(4-Carboxy-2-{4-carboxy-2-[(E)-3-...)
Affinity DataIC50:  5.50E+3nMAssay Description:Binding affinity to p60 src SH2 domain.More data for this Ligand-Target Pair
In DepthDetails Article
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