Affinity DataIC50: 0.600nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 2.10nMAssay Description:Tested for inhibitory activity against rat brain p21ras Ras Farnesyltransferase (FTase)More data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 21nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 40nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 48nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 52nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 56nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of CDK2/CyclinAMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:Inhibitory activity against alpha4-beta7/ MAdCAM integrin (mucosal addressin cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Rattus norvegicus)
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 80nMAssay Description:Tested for inhibitory activity against rat brain p21ras Ras Farnesyltransferase (FTase)More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of SHH in mouse C3H10T1/2 cells by Gli-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 82nMAssay Description:Inhibitory activity against alpha4-beta1 integrin (vascular cell adhesion molecule) in ELISA assayMore data for this Ligand-Target Pair
TargetIntegrin alpha-L/Integrin beta-2/Intercellular adhesion molecule 1(Homo sapiens (Human))
Genentech
Curated by ChEMBL
Genentech
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Inhibitory activity against association of LFA-1 with intercellular adhesion molecule 1More data for this Ligand-Target Pair