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Found 142 with Last Name = 'miura' and Initial = 'm'
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM31459(CHEMBL224485 | substituted biphenyl derivative, 21)
Affinity DataIC50:  89nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197327(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  150nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197325(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197331(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-({...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197330(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197324(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  590nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197326(2'-(3-carbamoyl-phenylcarbamoyl)-4-isobutylcarbamo...)
Affinity DataIC50:  690nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197329(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  860nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM31459(CHEMBL224485 | substituted biphenyl derivative, 21)
Affinity DataIC50:  880nMAssay Description:Inhibition of human Fxa by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030766(CHEMBL3342339)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of porcine tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197340(2'-({[4-(aminomethyl)phenyl]amino}carbonyl)-4-({[(...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTubulin beta chain(Sus scrofa)
Tokyo University Of Pharmacy And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50030765(NPI-2358 | Plinabulin)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of porcine tubulin polymerization by spectrophotometryMore data for this Ligand-Target Pair
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197336(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197341(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197333(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-[(...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197332(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}carb...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197334(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-[(...)
Affinity DataIC50:  4.20E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197338(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197339(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197335(2'-(3-Carbamoyl-phenylcarbamoyl)-4-isobutylcarbamo...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197328(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50:  9.10E+4nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025146(2-(4-Cyano-phenyl)-N-hydroxy-2-oxo-thioacetimidic ...)
Affinity DataIC50:  1.80E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII/Tissue factor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197337(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-({...)
Affinity DataIC50:  1.91E+5nMAssay Description:Inhibition of human TF/FVIIa complex by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197326(2'-(3-carbamoyl-phenylcarbamoyl)-4-isobutylcarbamo...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thrombin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM31459(CHEMBL224485 | substituted biphenyl derivative, 21)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thrombin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197327(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thrombin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197324(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human Fxa by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197325(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human Fxa by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197325(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thrombin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197324(4-({[(1S)-(aminocarbonyl)-3-methylbutyl]amino}-car...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human thrombin by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197326(2'-(3-carbamoyl-phenylcarbamoyl)-4-isobutylcarbamo...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human Fxa by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50197327(2'-({[3-(aminocarbonyl)phenyl]amino}carbonyl)-4-{[...)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human Fxa by chromogenic assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025141(2-(4-Bromo-phenyl)-N-hydroxy-2-oxo-thioacetimidic ...)
Affinity DataIC50:  2.10E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025142(CHEMBL46151 | N-Hydroxy-2-(4-methoxy-phenyl)-2-oxo...)
Affinity DataIC50:  2.60E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025131(2-(4-Chloro-phenyl)-N-hydroxy-2-oxo-thioacetimidic...)
Affinity DataIC50:  3.30E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50011780(2-[(E)-(hydroxyimino)methyl]-1-methylpyridinium ch...)
Affinity DataIC50:  3.40E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50020522(1-(((4-carbamoylpyridinium-1-yl)methoxy)methyl)-2-...)
Affinity DataIC50:  4.60E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025133(2-(4-Chloro-phenyl)-N-hydroxy-2-oxo-thioacetimidic...)
Affinity DataIC50:  5.20E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025130(2-(4-Bromo-phenyl)-N-hydroxy-2-oxo-thioacetimidic ...)
Affinity DataIC50:  7.10E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025127(CHEMBL416644 | Diethyl-{2-[2-(4-fluoro-phenyl)-N-h...)
Affinity DataIC50:  7.20E+5nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025143(CHEMBL297316 | {2-[2-(4-Fluoro-phenyl)-N-hydroxy-2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025145(CHEMBL296560 | {2-[2-(4-Bromo-phenyl)-N-hydroxy-2-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025144(CHEMBL47375 | {2-[N-Hydroxy-2-(4-methoxy-phenyl)-2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025136(CHEMBL556172 | N-Hydroxy-2-oxo-2-phenyl-thioacetim...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025135(CHEMBL296429 | [2-(N-Hydroxy-2-oxo-2-p-tolyl-aceti...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025134(2-(4-Chloro-phenyl)-N-hydroxy-2-oxo-thioacetimidic...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025138(CHEMBL296277 | {2-[2-(4-Cyano-phenyl)-N-hydroxy-2-...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025139(CHEMBL416464 | N-Hydroxy-2-(4-methoxy-phenyl)-2-ox...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025132(CHEMBL542609 | N-Hydroxy-2-oxo-2-p-tolyl-thioaceti...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50025128(CHEMBL296786 | {2-[2-(4-Chloro-phenyl)-N-hydroxy-2...)
Affinity DataIC50: >1.00E+6nMAssay Description:Reversible inhibition of Human AchEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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