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Found 42 with Last Name = 'moresco' and Initial = 'rm'
TargetAdenosine receptor A2a(Homo sapiens (Human))
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi:  0.0480nMAssay Description:Inhibitory activity against human adenosine A2A receptor expressed in HEK-293 cells by displacement of [3H]-SCH-58,261More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50176070(7-Methoxy-benzofuran-2-carboxylic acid {4-[4-(2,3-...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi:  0.5nMAssay Description:Inhibitory activity against adenosine A2A receptor in rat striatal membranes by displacement of [3H]-SCH-58,261More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50122041(1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3...)
Affinity DataKi:  0.600nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50137626(5-Bromo-N-{4-[4-(2,3-dichloro-phenyl)-piperazin-1-...)
Affinity DataKi:  2nMAssay Description:Binding affinity for rat dopamine D3 receptor using [11C]-GR-218,231More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50176070(7-Methoxy-benzofuran-2-carboxylic acid {4-[4-(2,3-...)
Affinity DataKi:  110nMAssay Description:Binding affinity for rat Alpha-1A adrenergic receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50176070(7-Methoxy-benzofuran-2-carboxylic acid {4-[4-(2,3-...)
Affinity DataKi:  180nMAssay Description:Binding affinity for rat Opioid receptor sigma 1 using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50176070(7-Methoxy-benzofuran-2-carboxylic acid {4-[4-(2,3-...)
Affinity DataKi:  184nMAssay Description:Binding affinity for rat 5-Hydroxytryptamine receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(RAT)
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50122041(1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3...)
Affinity DataKi:  342nMAssay Description:Binding affinity for rat Opioid receptor sigma 1 using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50176070(7-Methoxy-benzofuran-2-carboxylic acid {4-[4-(2,3-...)
Affinity DataKi:  373nMAssay Description:Binding affinity for rat dopamine D4 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50122041(1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3...)
Affinity DataKi:  575nMAssay Description:Binding affinity for rat 5-Hydroxytryptamine receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50176070(7-Methoxy-benzofuran-2-carboxylic acid {4-[4-(2,3-...)
Affinity DataKi:  720nMAssay Description:Binding affinity towards rat dopamine D2 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50122041(1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3...)
Affinity DataKi:  720nMAssay Description:Binding affinity towards rat dopamine D2 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(RAT)
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50122041(1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3...)
Affinity DataKi:  830nMAssay Description:Binding affinity for rat dopamine D4 receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi:  1.11E+3nMAssay Description:Inhibitory activity against human adenosine A1 receptor expressed in CHO cells by displacement of [3H]-DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi:  1.82E+3nMAssay Description:Displacement of [3H]-DPCPX from adenosine A1 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
University Of Milano/Bicocca

Curated by ChEMBL
LigandPNGBDBM50122041(1-Methoxy-naphthalene-2-carboxylic acid {4-[4-(2,3...)
Affinity DataKi:  5.10E+3nMAssay Description:Binding affinity for rat Alpha-1A adrenergic receptor using [11C] radiotracerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against human adenosine A2B receptor expressed in HEK-293 cells by displacement of [3H]-DPCPXMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Rattus norvegicus)
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against rat adenosine A3 receptor expressed in HEK-293 cells by displacement of [125I]-AB-MECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
University Of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50094037(2-Furan-2-yl-7-[3-(4-methoxy-phenyl)-propyl]-7H-py...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [125I]-AB-MECA from human adenosine A3 receptor expressed in HEK-293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140783(2-Hydroxymethyl-4-phenyl-quinoline-3-carboxylic ac...)
Affinity DataIC50:  0.000100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140770(2-Aminomethyl-4-phenyl-quinoline-3-carboxylic acid...)
Affinity DataIC50:  0.00170nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140773(2-Bromomethyl-4-phenyl-quinoline-3-carboxylic acid...)
Affinity DataIC50:  0.0100nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140785(2-Methylaminomethyl-4-phenyl-quinoline-3-carboxyli...)
Affinity DataIC50:  0.0110nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140786(4-Phenyl-quinoline-3-carboxylic acid (3,5-bis-trif...)
Affinity DataIC50:  0.0300nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140772(2-Methyl-4-phenyl-quinoline-3-carboxylic acid 3,5-...)
Affinity DataIC50:  0.0750nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  0.120nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140774(2-Dimethylaminomethyl-4-phenyl-quinoline-3-carboxy...)
Affinity DataIC50:  0.220nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140771(((2R,3R)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140776(2-Methyl-4-phenyl-quinoline-3-carboxylic acid (3,5...)
Affinity DataIC50:  3.10nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140788(2-Aminomethyl-4-phenyl-quinoline-3-carboxylic acid...)
Affinity DataIC50:  9nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140781(2-Methoxymethyl-4-phenyl-quinoline-3-carboxylic ac...)
Affinity DataIC50:  11nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140774(2-Dimethylaminomethyl-4-phenyl-quinoline-3-carboxy...)
Affinity DataIC50:  11nMAssay Description:Inhibition of labeled SP total binding against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells by the second binding componentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140782(2-Hydroxymethyl-4-phenyl-quinoline-3-carboxylic ac...)
Affinity DataIC50:  16nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140780(2-(tert-Butyl-dimethyl-silanyloxymethyl)-4-phenyl-...)
Affinity DataIC50:  17nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140779(2-Chloromethyl-4-phenyl-quinoline-3-carboxylic aci...)
Affinity DataIC50:  26nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140777(2-Bromomethyl-4-phenyl-quinoline-3-carboxylic acid...)
Affinity DataIC50:  52nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140787(2-[(Benzyl-methyl-amino)-methyl]-4-phenyl-quinolin...)
Affinity DataIC50:  180nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140775(4-Phenyl-quinoline-3-carboxylic acid 3,5-bis-trifl...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140778(2-(4-Methyl-piperazin-1-ylmethyl)-4-phenyl-quinoli...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140784(2-(1,3-Dioxo-1,3-dihydro-isoindol-2-ylmethyl)-4-ph...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells using [125I]- SP radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50140772(2-Methyl-4-phenyl-quinoline-3-carboxylic acid 3,5-...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibition of labeled SP total binding against human Tachykinin receptor 1 expressed in astrocytoma UC11MG cells by the second binding componentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed