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Found 31 with Last Name = 'nah' and Initial = 'sy'
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM82561(CAS_40796-97-2 | TROPANYL 3,5-DICHLOROBENZOATE | T...)
Affinity DataIC50:  770nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295828(3-(4-methoxybenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl...)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295834(3-(4-chlorobenzyl)-N-(3-morpholinopropyl)-2,4-diox...)
Affinity DataIC50:  1.30E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295826(3-(2-methoxybenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295824(3-(4-methoxyphenyl)-2,4-dioxo-N-(2-(piperidin-1-yl...)
Affinity DataIC50:  1.60E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196473(3-(4-fluorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295823(3-(4-fluorophenyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  1.90E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196475(3-(4-chlorobenzyl)-2,4-dioxo-N-(3-(piperidin-1-yl)...)
Affinity DataIC50:  1.95E+3nMAssay Description:Antagonist activity against T-type calcium channel alpha1GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295829(3-cyclohexyl-2,4-dioxo-N-(2-(piperidin-1-yl)ethyl)...)
Affinity DataIC50:  2.00E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196465(3-(4-chlorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  2.08E+3nMAssay Description:Antagonist activity against T-type calcium channel alpha1GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295825(3-(2-fluorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295832(3-(2-chlorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295830(2,4-dioxo-N-(2-(piperidin-1-yl)ethyl)-3-propyl-1,2...)
Affinity DataIC50:  2.20E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295831(3-methyl-2,4-dioxo-N-(2-(piperidin-1-yl)ethyl)-1,2...)
Affinity DataIC50:  2.20E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196469(3-(3-fluorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  2.40E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196478(3-(4-chlorobenzyl)-2,4-dioxo-N-(2-(pyrrolidin-1-yl...)
Affinity DataIC50:  2.46E+3nMAssay Description:Antagonist activity against T-type calcium channel alpha1GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295827(3-(3-methoxybenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl...)
Affinity DataIC50:  2.70E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295833(3-(4-chlorobenzyl)-N-(2-(2-methylpiperidin-1-yl)et...)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196465(3-(4-chlorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  3.30E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196480(3-(4-chlorobenzyl)-N-(2-(2-ethylpiperidin-1-yl)eth...)
Affinity DataIC50:  3.38E+3nMAssay Description:Antagonist activity against T-type calcium channel alpha1GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196466(3-(4-chlorobenzyl)-N-(3-(2-ethylpiperidin-1-yl)pro...)
Affinity DataIC50:  4.80E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196475(3-(4-chlorobenzyl)-2,4-dioxo-N-(3-(piperidin-1-yl)...)
Affinity DataIC50:  5.70E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295835(3-cyclohexyl-N-(3-(2-methylpiperidin-1-yl)propyl)-...)
Affinity DataIC50:  5.90E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196478(3-(4-chlorobenzyl)-2,4-dioxo-N-(2-(pyrrolidin-1-yl...)
Affinity DataIC50:  7.50E+3nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196473(3-(4-fluorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  9.23E+3nMAssay Description:Antagonist activity against T-type calcium channel alpha1GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196472(3-(4-chlorobenzyl)-N-(3-(2-methylpiperidin-1-yl)pr...)
Affinity DataIC50:  1.16E+4nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196480(3-(4-chlorobenzyl)-N-(2-(2-ethylpiperidin-1-yl)eth...)
Affinity DataIC50:  1.36E+4nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295822(3-(4-chlorobenzyl)-N-(2-morpholinoethyl)-2,4-dioxo...)
Affinity DataIC50:  1.58E+4nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent T-type calcium channel subunit alpha-1G(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50196469(3-(3-fluorobenzyl)-2,4-dioxo-N-(2-(piperidin-1-yl)...)
Affinity DataIC50:  1.69E+4nMAssay Description:Antagonist activity against T-type calcium channel alpha1GMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295838(3-(4-fluorobenzyl)-N-(2-morpholinoethyl)-2,4-dioxo...)
Affinity DataIC50:  1.98E+4nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Konkuk University

Curated by ChEMBL
LigandPNGBDBM50295837(3-(4-fluorophenyl)-N-(2-morpholinoethyl)-2,4-dioxo...)
Affinity DataIC50:  5.70E+4nMAssay Description:Antagonist activity at 5HT3A receptor expressed in Xenopus oocyteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed