TargetLong-chain-fatty-acid--AMP ligase FadD32(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataIC50: 7.70E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis FAAL32 using AMPC12 as substrate incubated for 50 mins and measured by spectrophotometric assayMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 385nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 13nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 52nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 42nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 0.700nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 33nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 45nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 388nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 336nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 271nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 101nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 217nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 515nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: >5.00E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 1.46E+3nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 197nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 340nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 376nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 428nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 176nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 809nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 8.04nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 8.05nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 157nMAssay Description:Protection of human pregnane X receptor against proteolytic digestion in presence of trypsinMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 49nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
University Of Montpellier
Curated by ChEMBL
University Of Montpellier
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:Agonist activity at human pregnane X receptor expressed in HGPXR reporter cellsMore data for this Ligand-Target Pair