Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of glycogen phosphorylase in rat hepatocytes assessed as reduction in basal glycogenolysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of glycogen phosphorylase in rat hepatocytes assessed as reduction in glucagom-induced glycogenolysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.39E+3nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.85E+3nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.38E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.53E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 12386-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.39E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.67E+5nMAssay Description:Binding affinity to PBP2a in methicillin-resistant Staphylococcus aureus 123-1 by [14C]benzylpenicillin labelled competitive assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 400nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 54nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 25nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 90nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.5nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 35nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.40nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.5nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 5.40nMAssay Description:Agonist activity at human S1P1 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: >2.00E+4nMAssay Description:Agonist activity at human S1P3 receptor by [S35]GTPgammaS binding assayMore data for this Ligand-Target Pair