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Found 17 with Last Name = 'namboodiri' and Initial = 'v'
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM13336(4-[4-(4-fluorophenyl)-2-(4-methanesulfinylphenyl)-...)
Affinity DataIC50:  290nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174086(CHEMBL198470 | N-(3-hydroxy-4-(1-hydroxy-2-methylp...)
Affinity DataIC50:  400nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174085(CHEMBL198563 | N-(3-(trifluoromethyl)benzyl)-4-phe...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174095(CHEMBL198832 | N-(3-(trifluoromethoxy)benzyl)-4-ph...)
Affinity DataIC50:  600nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174098(CHEMBL197228 | N-((2,3-dihydro-1H-inden-5-yl)methy...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174090(CHEMBL199074 | N-(4-(trifluoromethyl)benzyl)-4-phe...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174097(4-phenoxy-N-(pyridin-2-ylmethyl)benzamide | CHEMBL...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174096(CHEMBL199174 | N-(4-methyl-benzyl)-4-phenoxy-benza...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174092(CHEMBL199229 | N-(3-hydroxy-4-(1-hydroxy-2-methylp...)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174088(4-(2-hydroxybenzylamino)-N-(3-(4-fluorophenoxy)phe...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174100(4-(2-hydroxybenzylamino)-N-(3-(2,4-difluorophenoxy...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174089(4-(2-hydroxybenzylamino)-N-(3-phenoxyphenyl)piperi...)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174099(2-((1-(3-phenoxybenzylsulfonyl)piperidin-4-ylamino...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174094(4-(2-hydroxybenzylamino)-N-(3-(2-chlorophenoxy)phe...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174091(4-(benzylamino)-N-(3-phenoxyphenyl)piperidine-1-su...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174087(4-(naphthalen-1-ylmethylamino)-N-(3-phenoxyphenyl)...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
Locus Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50174093(4-(2-hydroxybenzylamino)-N-(3-(3-(trifluoromethyl)...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against p38alpha MAPKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed