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Found 59 with Last Name = 'nawano' and Initial = 'm'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543892(CHEMBL4649482)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543890(CHEMBL4641678)
Affinity DataIC50:  1.67E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543895(CHEMBL4646396)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543889(CHEMBL4645293)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543894(CHEMBL4637653)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543893(CHEMBL4632835)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Chiba University

Curated by ChEMBL
LigandPNGBDBM50543896(CHEMBL4644080)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161677(4-[3-(5-Chloro-thiazol-2-yl)-1-cyclopentylmethyl-u...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161675(3-(5-Chloro-thiazol-2-yl)-1-(4-methanesulfonyl-phe...)
Affinity DataEC50:  6.80E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161680(3-(5-Chloro-thiazol-2-yl)-1-furan-2-ylmethyl-1-(4-...)
Affinity DataEC50:  1.15E+4nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161681(3-(5-Chloro-thiazol-2-yl)-1-(6-cyano-pyridin-3-yl)...)
Affinity DataEC50:  7.70E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161682(3-(5-Chloro-thiazol-2-yl)-1-cyclopentylmethyl-1-(3...)
Affinity DataEC50:  1.40E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161678(3-(5-Chloro-thiazol-2-yl)-1-cyclopentylmethyl-1-(6...)
Affinity DataEC50:  2.70E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161679(3-(5-Chloro-thiazol-2-yl)-1-(4-cyano-phenyl)-1-cyc...)
Affinity DataEC50:  2.40E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161684(1-Cyclopentylmethyl-3-(6-methanesulfonyl-benzothia...)
Affinity DataEC50:  3.29E+4nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161685(1-Cyclopentylmethyl-1-(6-methoxy-pyridin-3-yl)-3-t...)
Affinity DataEC50:  1.92E+4nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161683(3-(5-Chloro-thiazol-2-yl)-1-(4-methanesulfonyl-phe...)
Affinity DataEC50:  4.90E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161674(3-Cyclopentyl-2-(4-methanesulfonyl-phenyl)-N-thiaz...)
Affinity DataEC50:  2.20E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161686(3-(5-Chloro-thiazol-2-yl)-1-cyclopentylmethyl-1-(4...)
Affinity DataEC50:  1.30E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161687(3-(5-Chloro-thiazol-2-yl)-1-cyclopentylmethyl-1-(4...)
Affinity DataEC50:  1.50E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161688(3-(5-Chloro-thiazol-2-yl)-1-(4-methanesulfonyl-phe...)
Affinity DataEC50:  6.60E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161689(3-(5-Chloro-thiazol-2-yl)-1-(4-methanesulfonyl-phe...)
Affinity DataEC50:  2.19E+4nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161690(3-(5-Chloro-thiazol-2-yl)-1-cyclopentylmethyl-1-(3...)
Affinity DataEC50:  2.60E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161691(CHEMBL180172 | N-{3-[3-(5-Chloro-thiazol-2-yl)-1-c...)
Affinity DataEC50:  300nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161694(3-(5-Bromo-thiazol-2-yl)-1-(4-methanesulfonyl-phen...)
Affinity DataEC50:  6.50E+3nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161693(3-(5-Chloro-thiazol-2-yl)-1-(4-methanesulfonyl-phe...)
Affinity DataEC50:  2.16E+4nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161668(1-Cyclopentylmethyl-1-(4-methanesulfonyl-phenyl)-3...)
Affinity DataEC50:  9.70E+3nMAssay Description:Effective concentration for glucokinase activation with 15 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161695(1-(4-Bromo-3-fluoro-phenyl)-3-(5-chloro-thiazol-2-...)
Affinity DataEC50:  700nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Rattus norvegicus)
Osi Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50161692(1-(3-Chloro-4-methyl-phenyl)-3-(5-chloro-thiazol-2...)
Affinity DataEC50:  400nMAssay Description:Effective concentration for glucokinase activation with 5 mM glucoseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251802((E)-2-phenyl-N-(pyrazin-2-yl)-3-(thiophen-2-yl)acr...)
Affinity DataEC50:  2.60E+4nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251450((R)-2-(4-(cyclopentylsulfonyl)phenyl)-N-(5-fluorot...)
Affinity DataEC50:  70nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251421((R)-2-(4-(cyclobutylsulfonyl)phenyl)-N-(5-fluoroth...)
Affinity DataEC50:  140nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251392((R)-N-(5-fluorothiazol-2-yl)-2-(4-(methylsulfonyl)...)
Affinity DataEC50:  1.43E+3nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251391((2R)-2-(4-Cyclopropanesulfonylphenyl)-N-(5-fluorot...)
Affinity DataEC50:  130nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251390((R)-2-(4-(cyclopropylsulfonyl)phenyl)-N-(5-methylt...)
Affinity DataEC50:  580nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251389((R)-2-(4-(cyclopropylsulfonyl)phenyl)-3-(tetrahydr...)
Affinity DataEC50:  570nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251388((S)-2-(4-(methylsulfonyl)phenyl)-3-(tetrahydro-2H-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251833((R)-2-(4-(methylsulfonyl)phenyl)-3-(tetrahydro-2H-...)
Affinity DataEC50:  3.47E+3nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251832(2-(4-(methylsulfonyl)phenyl)-3-(tetrahydro-2H-pyra...)
Affinity DataEC50:  8.93E+3nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251831(2-(4-(methylsulfonyl)phenyl)-3-(tetrahydro-2H-pyra...)
Affinity DataEC50:  2.30E+3nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251830((Z)-2-(4-(methylsulfonyl)phenyl)-N-(thiazol-2-yl)-...)
Affinity DataEC50:  560nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50251829(2-phenyl-N-(thiazol-2-yl)-3-(thiophen-2-yl)acrylam...)
Affinity DataEC50:  1.08E+4nMAssay Description:Activation of GST fused human liver glucokinase assessed as generation of NADPH by G6PDH coupled assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543888(CHEMBL4641724)
Affinity DataEC50:  5.60E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543889(CHEMBL4645293)
Affinity DataEC50:  420nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543890(CHEMBL4641678)
Affinity DataEC50:  41nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543891(CHEMBL4638344)
Affinity DataEC50:  2.40E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543892(CHEMBL4649482)
Affinity DataEC50:  160nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543893(CHEMBL4632835)
Affinity DataEC50:  220nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543894(CHEMBL4637653)
Affinity DataEC50:  1.17E+3nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHexokinase-4(Homo sapiens (Human))
(Osi) Prosidion

Curated by ChEMBL
LigandPNGBDBM50543895(CHEMBL4646396)
Affinity DataEC50:  700nMAssay Description:Activation of human glucokinaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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