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Found 14 with Last Name = 'neame' and Initial = 'sj'
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173167((S)-(2-(4-fluorophenyl)-3-(2-(propylamino)pyrimidi...)
Affinity DataIC50:  2.5nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173169(CHEMBL383799 | [(R)-2-(4-Fluoro-phenyl)-3-(2-propy...)
Affinity DataIC50:  3nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173173(CHEMBL383348 | {4-[(S)-2-(4-Fluoro-phenyl)-5-(4-me...)
Affinity DataIC50:  10.9nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173167((S)-(2-(4-fluorophenyl)-3-(2-(propylamino)pyrimidi...)
Affinity DataIC50:  28nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173169(CHEMBL383799 | [(R)-2-(4-Fluoro-phenyl)-3-(2-propy...)
Affinity DataIC50:  31nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173166(CHEMBL371720 | N-{3-[4-(3-Azido-phenyl)-5-pyridin-...)
Affinity DataIC50:  46nMAssay Description:Inhibitory concentration against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173173(CHEMBL383348 | {4-[(S)-2-(4-Fluoro-phenyl)-5-(4-me...)
Affinity DataIC50:  54nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173168(4-[(S)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)
Affinity DataIC50:  61.2nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173172(4-[(R)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)
Affinity DataIC50:  116nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173171(CHEMBL199247 | N-(3-(4-(4-fluorophenyl)-5-(pyridin...)
Affinity DataIC50:  130nMAssay Description:Inhibitory concentration against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173170(CHEMBL198261 | {4-[(R)-2-(4-Fluoro-phenyl)-5-(4-me...)
Affinity DataIC50:  217nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173170(CHEMBL198261 | {4-[(R)-2-(4-Fluoro-phenyl)-5-(4-me...)
Affinity DataIC50:  233nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173172(4-[(R)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)
Affinity DataIC50:  270nMAssay Description:Inhibitory activity against c-Jun N-terminal kinase 3 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
University College London

Curated by ChEMBL
LigandPNGBDBM50173168(4-[(S)-2-(4-Fluoro-phenyl)-5-(4-methoxy-benzyloxym...)
Affinity DataIC50:  295nMAssay Description:Inhibitory activity against p38 at a concentration of 1.0 uM More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed