TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 0.160nMAssay Description:Enzyme inhibitory activity towards Angiotensin I converting enzymeMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 4nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 23nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cortices and cerebella by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 32nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 46nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 50nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 62nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 64nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 67nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 69nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 95nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 109nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 141nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 188nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 189nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 209nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 209nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cortices and cerebella by competition binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 215nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 229nMAssay Description:Binding affinity of the compound towards Opioid receptor delta 1 was determined using [d-Ser2, Leu5, Thr6] enkephalin (DSLET) as the radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 236nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 246nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 254nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 316nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 333nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 338nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 392nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 393nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 406nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 430nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 435nMAssay Description:Binding affinity for [3H]- pentazocine at sigma opioid receptorMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 547nMAssay Description:Binding affinity of the compound towards Opioid receptor mu 1 was determined using ([d-Ala2,MePhe4, Gly5-ol]-enkephalin (DAMGO) as the radioligand.More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 552nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 566nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 605nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 642nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cortices and cerebella by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 721nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 740nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membrane by liquid scintillation counting analysisMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Torrey Pines Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 767nMAssay Description:Displacement of [3H]U69593 from kappa opioid receptor in guinea pig cortices and cerebella by competition binding assayMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Institute For Molecular Studies
Curated by ChEMBL
Institute For Molecular Studies
Curated by ChEMBL
Affinity DataKi: 878nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat cortices by competition binding assayMore data for this Ligand-Target Pair