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Found 35 with Last Name = 'nelson' and Initial = 'gl'
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092069(CHEMBL3582422 | US9296728, 20)
Affinity DataIC50:  8nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092072(CHEMBL3582419 | US9296728, 14)
Affinity DataIC50:  9nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092058(CHEMBL3582408)
Affinity DataIC50:  10nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092068(CHEMBL3582423)
Affinity DataIC50:  11nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092071(CHEMBL3582420 | US9296728, 18)
Affinity DataIC50:  11nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092073(CHEMBL3582418 | US9296728, 13)
Affinity DataIC50:  12nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092065(CHEMBL3582426)
Affinity DataIC50:  25nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092067(CHEMBL3582424 | US9296728, 16)
Affinity DataIC50:  29nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092076(CHEMBL3582415)
Affinity DataIC50:  30nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092057(CHEMBL3582409 | US9296728, 4)
Affinity DataIC50:  30nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092070(CHEMBL3582421 | US9296728, 15)
Affinity DataIC50:  34nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092066(CHEMBL3582425)
Affinity DataIC50:  48nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092059(CHEMBL3582407)
Affinity DataIC50:  70nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092075(CHEMBL3582416 | US9296728, 11)
Affinity DataIC50:  70nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM214702(US9296728, 25)
Affinity DataIC50:  90nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092018(CHEMBL3582410 | US9296728, 9)
Affinity DataIC50:  100nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092078(CHEMBL3582413 | US9296728, 7)
Affinity DataIC50:  110nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM4345((2E)-2-cyano-3-[4-(dimethylamino)phenyl]prop-2-eno...)
Affinity DataIC50:  140nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092017(CHEMBL3582411 | US9296728, 5)
Affinity DataIC50:  140nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092074(CHEMBL3582417 | US9296728, 12)
Affinity DataIC50:  140nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM214700(US9296728, 23)
Affinity DataIC50:  170nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM214701(US9296728, 24)
Affinity DataIC50:  210nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50442702(CHEMBL2442511 | US9296728, 26)
Affinity DataIC50:  380nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092077(CHEMBL3582414 | US9296728, 8)
Affinity DataIC50:  400nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM214699(US9296728, 22)
Affinity DataIC50:  450nMAssay Description:Inhibition of MCT1 in rat brain endothelial 4 cells assessed as L-[14C]-Lactate Uptake after 15 mins by scintillation spectrometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM4343((2E)-2-cyano-3-(4-methoxyphenyl)prop-2-enoic acid ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092060(CHEMBL3582406)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM4347((2E)-2-cyano-3-(4-nitrophenyl)prop-2-enoic acid | ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092061(CHEMBL3582405)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092062(CHEMBL3582404)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM4346((2E)-2-cyano-3-(4-methylphenyl)prop-2-enoic acid |...)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM4344((2E)-2-cyano-3-(4-fluorophenyl)prop-2-enoic acid |...)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092063(CHEMBL3582403)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092064(CHEMBL3582402)
Affinity DataIC50:  500nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonocarboxylate transporter 1(Rattus norvegicus (Rat))
Medical School Duluth

Curated by ChEMBL
LigandPNGBDBM50092016(CHEMBL3582412 | US9296728, 6)
Affinity DataIC50:  880nMAssay Description:Inhibition of MCT1-mediated lactate transport in rat RBE4 cells incubated for 15 mins by [14C]-lactate uptake assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed