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Found 193 with Last Name = 'neubig' and Initial = 'rr'
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  0.620nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  0.780nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  1.04nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  1.57nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  1.78nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  3.02nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81444(CAS_185453 | NSC_185453 | WB 4101 | WB-4101)
Affinity DataKi:  3.18nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  3.71nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  3.76nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50019492((+)2-(2-Methoxy-2,3-dihydro-benzo[1,4]dioxin-2-yl)...)
Affinity DataKi:  3.83nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  4.59nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM82520(BRL44408 | CAS_121850 | NSC_121850)
Affinity DataKi:  5.68nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM30712(6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimet...)
Affinity DataKi:  9.68nMMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50013515((+)-yohimbine | (16alpha,17alpha)-17-hydroxyyohimb...)
Affinity DataKi:  13.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81444(CAS_185453 | NSC_185453 | WB 4101 | WB-4101)
Affinity DataKi:  14.6nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81772(ARC-239 | CAS_122211 | NSC_122211)
Affinity DataKi:  19.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81772(ARC-239 | CAS_122211 | NSC_122211)
Affinity DataKi:  31.8nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM30712(6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimet...)
Affinity DataKi:  35.5nMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81984(CAS_29110-47-2 | Guanfacine | NSC_3519)
Affinity DataKi:  50.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50262179(Iodoclonidine-p | p-iodoclonidine)
Affinity DataKi:  51.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50020192(8-(2,3-Dihydro-benzo[1,4]dioxin-2-ylmethyl)-1-phen...)
Affinity DataKi:  54.3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  57.2nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81979(CAS_5051-62-7 | CAS_65636 | Fluprofylline | Guanab...)
Affinity DataKi:  57.5nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81444(CAS_185453 | NSC_185453 | WB 4101 | WB-4101)
Affinity DataKi:  78nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-1,3-diazacyclopentene-(2) ...)
Affinity DataKi:  85.1nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  116nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM82519(4-amino-5-chloro-2-methoxy-N-(8-methyl-8-azabicycl...)
Affinity DataKi:  150nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM30712(6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimet...)
Affinity DataKi:  185nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81926(Aminoclonidine, p | CAS_66711-21-5 | NSC_51763 | p...)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM34572(BRIMONIDINE | CHEMBL844 | MLS000069370 | SMR000058...)
Affinity DataKi:  479nMMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM84342(4-[1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol...)
Affinity DataKi:  646nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM82520(BRL44408 | CAS_121850 | NSC_121850)
Affinity DataKi:  651nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81984(CAS_29110-47-2 | Guanfacine | NSC_3519)
Affinity DataKi:  1.02E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM81984(CAS_29110-47-2 | Guanfacine | NSC_3519)
Affinity DataKi:  1.12E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM29568(CHEMBL2 | PRAZOSIN | PRAZOSIN HYDROCHLORIDE | [3H]...)
Affinity DataKi:  2.25E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM30712(6-tert-butyl-3-(2-imidazolin-2-ylmethyl)-2,4-dimet...)
Affinity DataKi:  2.98E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM50027069((2,6-Dimethyl-phenyl)-[1,3]thiazinan-2-ylidene-ami...)
Affinity DataKi:  3.16E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM35234(DL-[7-3H]norepinephrine | NOREPINEPHRINE | Noradre...)
Affinity DataKi:  5.62E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM85676(BHT-933 | CAS_128-37-0 | NSC_169743)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAlpha-2A adrenergic receptor(PIG)
University Of Michigan

Curated by PDSP Ki Database
LigandPNGBDBM25392(4-[1-hydroxy-2-(isopropylamino)ethyl]pyrocatechol;...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384752(CHEMBL2037351)
Affinity DataIC50:  5.40nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384751(CHEMBL2037350)
Affinity DataIC50:  7.20nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384755(CHEMBL2037352)
Affinity DataIC50:  8.60nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384777(CHEMBL2037229)
Affinity DataIC50:  11nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384754(CHEMBL2037234)
Affinity DataIC50:  13nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384767(CHEMBL2037365)
Affinity DataIC50:  14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM7779(4-butyl-2-ethyl-1,2,4-thiadiazolidine-3,5-dione | ...)
Affinity DataIC50:  14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384776(CHEMBL2037228)
Affinity DataIC50:  14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384743(CHEMBL2037235)
Affinity DataIC50:  14nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRegulator of G-protein signaling 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384757(CHEMBL2037354)
Affinity DataIC50:  15nMAssay Description:Inhibition of RGS4 interaction with Galpha0 protein by flow cytometry protein interaction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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