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Found 27 with Last Name = 'newcomb' and Initial = 'lf'
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50009073(4-(5-cyclopentyloxycarbonylamino-1-methyl-1H-indol...)
Affinity DataKi:  0.340nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041356(1-Ethyl-3-[2-methoxy-4-(toluene-2-sulfonylaminocar...)
Affinity DataKi:  0.380nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041349(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  0.420nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041357(1-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  0.440nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041344(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  0.570nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041336(3-[4-(2-Chloro-benzenesulfonylaminocarbonyl)-2-met...)
Affinity DataKi:  0.570nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041350(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  1.20nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041352(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  1.30nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041339(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  1.5nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041353(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  1.70nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041348(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  2.10nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041360(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  2.20nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041337(3-[4-(2-Bromo-benzenesulfonylaminocarbonyl)-2-meth...)
Affinity DataKi:  2.40nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50000817(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  3.20nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041345(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  3.80nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041340(1-[4-(2-Chloro-benzenesulfonylaminocarbonyl)-2-met...)
Affinity DataKi:  4.20nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041347(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  4.60nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041341(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  4.70nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041355(1-[4-(2-Chloro-benzenesulfonylaminocarbonyl)-2-met...)
Affinity DataKi:  4.90nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041338(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  5nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041342(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  5.20nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041351(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  5.30nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041343(1-Ethyl-3-[2-methoxy-4-(toluene-2-sulfonylaminocar...)
Affinity DataKi:  5.30nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041346(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  7.30nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041354(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  7.5nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041358(1-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  7.70nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCysteinyl leukotriene receptor 1(GUINEA PIG)
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50041359(3-[2-Methoxy-4-(toluene-2-sulfonylaminocarbonyl)-b...)
Affinity DataKi:  12nMAssay Description:Inhibition constant for displacement of [3H]-LTD4 on guinea pig lung parenchymal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed