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Found 68 with Last Name = 'nibbio' and Initial = 'm'
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592391(CHEMBL5187766)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592384(CHEMBL5195846)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50441357(CHEMBL2431805)
Affinity DataIC50:  4nMAssay Description:Inhibition of GST-tagged Tankyrases 2 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592392(CHEMBL5193402)
Affinity DataIC50:  5.20nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592390(CHEMBL5172085)
Affinity DataIC50:  5.70nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)
Affinity DataIC50:  5.80nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
TargetPoly [ADP-ribose] polymerase tankyrase-1(Homo sapiens (Human))
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50441357(CHEMBL2431805)
Affinity DataIC50:  11nMAssay Description:Inhibition of GST-tagged Tankyrases 1 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592390(CHEMBL5172085)
Affinity DataIC50:  16nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592395(CHEMBL5183771)
Affinity DataIC50:  18nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592391(CHEMBL5187766)
Affinity DataIC50:  25nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592384(CHEMBL5195846)
Affinity DataIC50:  26nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetIntegrase(Human immunodeficiency virus 1)
Irbm

Curated by ChEMBL
LigandPNGBDBM25351(N-[2-(4-{[(4-fluorophenyl)methyl]carbamoyl}-5-hydr...)
Affinity DataIC50:  27nMAssay Description:Inhibition of wild type recombinant HIV1 His6-tagged integrase expressed in Escherichia coli BL21 using 18 nucleotide 3'-biotin labeled DNA acceptor ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592394(CHEMBL5199280)
Affinity DataIC50:  29nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592395(CHEMBL5183771)
Affinity DataIC50:  54nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592391(CHEMBL5187766)
Affinity DataIC50:  55nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592378(CHEMBL5188089)
Affinity DataIC50:  62nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592392(CHEMBL5193402)
Affinity DataIC50:  64nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592376(CHEMBL5177309)
Affinity DataIC50:  77nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592386(CHEMBL5189772)
Affinity DataIC50:  97nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592394(CHEMBL5199280)
Affinity DataIC50:  110nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50446376(CHEMBL3109630)
Affinity DataIC50:  118nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592377(CHEMBL5194471)
Affinity DataIC50:  206nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592386(CHEMBL5189772)
Affinity DataIC50:  252nMAssay Description:Inhibition of G9a (unknown origin) assessed as effect on H3K9 methylation by cell based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592384(CHEMBL5195846)
Affinity DataIC50:  328nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592392(CHEMBL5193402)
Affinity DataIC50:  332nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592390(CHEMBL5172085)
Affinity DataIC50:  404nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592381(CHEMBL5185925)
Affinity DataIC50:  440nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592393(CHEMBL5202307)
Affinity DataIC50:  480nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592385(CHEMBL5184153)
Affinity DataIC50:  628nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592379(CHEMBL5191627)
Affinity DataIC50:  633nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592387(CHEMBL5191130)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592389(CHEMBL5209060)
Affinity DataIC50:  1.08E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592388(CHEMBL5207069)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592394(CHEMBL5199280)
Affinity DataIC50:  1.11E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592386(CHEMBL5189772)
Affinity DataIC50:  1.95E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592395(CHEMBL5183771)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592377(CHEMBL5194471)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPoly [ADP-ribose] polymerase tankyrase-2(Homo sapiens (Human))
Siena Biotech

Curated by ChEMBL
LigandPNGBDBM50082111(CHEMBL3422630)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of GST-tagged Tankyrases 2 (unknown origin) by autoPARsylationassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592378(CHEMBL5188089)
Affinity DataIC50:  3.46E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592385(CHEMBL5184153)
Affinity DataIC50:  4.37E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592381(CHEMBL5185925)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592382(CHEMBL5191872)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592383(CHEMBL5198356)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592379(CHEMBL5191627)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592380(CHEMBL5183788)
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of G9a (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592376(CHEMBL5177309)
Affinity DataIC50:  5.23E+3nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592388(CHEMBL5207069)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592393(CHEMBL5202307)
Affinity DataIC50:  1.55E+4nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetHistone-lysine N-methyltransferase EHMT1(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50592387(CHEMBL5191130)
Affinity DataIC50:  1.56E+4nMAssay Description:Inhibition of GLP (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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