Affinity DataKi: 0.112nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.143nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.203nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.222nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.286nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 0.960nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
Target3-beta-hydroxysteroid-Delta(8),Delta(7)-isomerase(Homo sapiens (Human))
Stanford University
Curated by ChEMBL
Stanford University
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity to EBPMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat liver homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Displacement of [3H](+)-pentazocine from Sigma1 receptor in rat brain homogenateMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 6.40nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 180nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 400nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: 2.10E+3nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Vrije Universiteit Brussel
Curated by ChEMBL
Vrije Universiteit Brussel
Curated by ChEMBL
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 1.90E+4nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 3.98E+4nMAssay Description:Affinity fo the compound against human Intestinal peptide transporter PepT1 in Caco-2 cells was measured as inhibition of [14C]-Gly-Sar uptakeMore data for this Ligand-Target Pair
Affinity DataKi: 6.80E+4nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 1.33E+5nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 2.10E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.80E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in Caco-2 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.17E+5nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 9.05E+5nMAssay Description:Affinity for hPEPT1 in mature Caco-2 cell monolayers using [14C]-Gly-SarMore data for this Ligand-Target Pair
Affinity DataKi: 4.68E+7nMAssay Description:Binding affinity to PEPT1 in human Caco2 cells assessed as inhibition of [14C]Gly-Sar apical uptake after 5 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+8nMAssay Description:Binding affinity to PEPT1 in human Caco2 cells assessed as inhibition of [14C]Gly-Sar apical uptake after 5 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.45E+8nMAssay Description:Binding affinity to PEPT1 in human Caco2 cells assessed as inhibition of [14C]Gly-Sar apical uptake after 5 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.51E+8nMAssay Description:Binding affinity to PEPT1 in human Caco2 cells assessed as inhibition of [14C]Gly-Sar apical uptake after 5 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 2.57E+8nMAssay Description:Binding affinity to PEPT1 in human Caco2 cells assessed as inhibition of [14C]Gly-Sar apical uptake after 5 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 3.24E+8nMAssay Description:Binding affinity to PEPT1 in human Caco2 cells assessed as inhibition of [14C]Gly-Sar apical uptake after 5 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.350nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 0.660nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Agonist activity at mu opioid receptor in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 2.80nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataIC50: 4nMAssay Description:Antagonist activity at human CRTH2 receptor assessed as inhibition of PGD2-induced signaling by inositol-phosphate assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.90nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at FPR2 in human peripheral blood polymorphonuclear neutrophils assessed as inhibition of WKYMVM-peptide induced ROS production p...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at FPR2 in human peripheral blood polymorphonuclear neutrophils assessed as inhibition of WKYMVM-peptide induced ROS production p...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at FPR2 in human peripheral blood polymorphonuclear neutrophils assessed as inhibition of WKYMVM-peptide induced ROS production p...More data for this Ligand-Target Pair