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Found 365 with Last Name = 'nienaber' and Initial = 'v'
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147093(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  0.620nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147096(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  2nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147095(6-Carbamimidoyl-4-(5-ethanesulfonyl-furan-3-yl)-na...)
Affinity DataKi:  2.10nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147095(6-Carbamimidoyl-4-(5-ethanesulfonyl-furan-3-yl)-na...)
Affinity DataKi:  3nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147091(6-Carbamimidoyl-4-(5-ethanesulfonyl-furan-3-yl)-na...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157087(6-(2-Phenyl-cyclopropyl)-8-(pyrimidin-2-ylamino)-n...)
Affinity DataKi:  5nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138673(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-e...)
Affinity DataKi:  6.30nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147089(6-Carbamimidoyl-4-(tetrahydro-furan-3-yl)-naphthal...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157094(8-(Pyrimidin-2-ylamino)-6-((E)-styryl)-naphthalene...)
Affinity DataKi:  10nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138676(6-Carbamimidoyl-naphthalene-2-carboxylic acid (3-c...)
Affinity DataKi:  11nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147094(6-Carbamimidoyl-4-(5-ethylsulfanyl-furan-3-yl)-nap...)
Affinity DataKi:  11nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147089(6-Carbamimidoyl-4-(tetrahydro-furan-3-yl)-naphthal...)
Affinity DataKi:  12nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138661(6-Carbamimidoyl-naphthalene-2-carboxylic acid (3,5...)
Affinity DataKi:  13nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138656(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1,2...)
Affinity DataKi:  16.5nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147091(6-Carbamimidoyl-4-(5-ethanesulfonyl-furan-3-yl)-na...)
Affinity DataKi:  18nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147091(6-Carbamimidoyl-4-(5-ethanesulfonyl-furan-3-yl)-na...)
Affinity DataKi:  19nMAssay Description:Binding affinity towards P-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147093(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  20nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138676(6-Carbamimidoyl-naphthalene-2-carboxylic acid (3-c...)
Affinity DataKi:  22nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138665(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-i...)
Affinity DataKi:  23.5nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138658(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-c...)
Affinity DataKi:  26.5nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138661(6-Carbamimidoyl-naphthalene-2-carboxylic acid (3,5...)
Affinity DataKi:  28nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138674(6-Carbamimidoyl-naphthalene-2-carboxylic acid (3-c...)
Affinity DataKi:  28nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157093(6-[2-(1-Cyclohexyl-2-methyl-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  28nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157098(6-[2-((S)-1-Isopropyl-3,4-dihydro-isoquinolin-7-yl...)
Affinity DataKi:  30nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147084(6-Carbamimidoyl-4-(tetrahydro-furan-3-yl)-naphthal...)
Affinity DataKi:  30nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157093(6-[2-(1-Cyclohexyl-2-methyl-1,2,3,4-tetrahydro-iso...)
Affinity DataKi:  31nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147086(8-(PYRIMIDIN-2-YLAMINO)NAPHTHALENE-2-CARBOXIMIDAMI...)
Affinity DataKi:  35nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138668(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-c...)
Affinity DataKi:  35.5nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138666(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-h...)
Affinity DataKi:  38nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147095(6-Carbamimidoyl-4-(5-ethanesulfonyl-furan-3-yl)-na...)
Affinity DataKi:  38nMAssay Description:Binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138658(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-c...)
Affinity DataKi:  39nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147094(6-Carbamimidoyl-4-(5-ethylsulfanyl-furan-3-yl)-nap...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards Urokinase-type plasminogen activator (urokinase)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147096(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  40nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147093(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  40nMAssay Description:Binding affinity towards P-kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138662(6-Carbamimidoyl-naphthalene-2-carboxylic acid (4-a...)
Affinity DataKi:  40nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
TargetTrypsin(Sus scrofa)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147096(6-Carbamimidoyl-4-(pyrimidin-2-ylamino)-naphthalen...)
Affinity DataKi:  40nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157094(8-(Pyrimidin-2-ylamino)-6-((E)-styryl)-naphthalene...)
Affinity DataKi:  42nMAssay Description:Binding affinity value against kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138667(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-i...)
Affinity DataKi:  42nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138665(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-i...)
Affinity DataKi:  43nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147088(6-Carbamimidoyl-4-furan-3-yl-naphthalene-2-carboxy...)
Affinity DataKi:  45nMAssay Description:Binding affinity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147088(6-Carbamimidoyl-4-furan-3-yl-naphthalene-2-carboxy...)
Affinity DataKi:  45nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157090(6-(2-(1-isopropyl-2-methyl-1,2,3,4-tetrahydroisoqu...)
Affinity DataKi:  47nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157083(6-Phenethyl-8-(pyrimidin-2-ylamino)-naphthalene-2-...)
Affinity DataKi:  47nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138667(6-Carbamimidoyl-naphthalene-2-carboxylic acid (1-i...)
Affinity DataKi:  48nMAssay Description:Binding affinity to human urokinase-type plasminogen activator (microPa).More data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157092(6-[2-(1-Cyclohexyl-3,4-dihydro-isoquinolin-7-yl)-c...)
Affinity DataKi:  50nMAssay Description:Binding affinity value against urokinase plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50138671(6-Carbamimidoyl-naphthalene-2-carboxylic acid (3-i...)
Affinity DataKi:  51nMAssay Description:Binding affinity against porcine trypsin was determined.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50147094(6-Carbamimidoyl-4-(5-ethylsulfanyl-furan-3-yl)-nap...)
Affinity DataKi:  53nMAssay Description:Binding affinity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157096(6-(2-(1-isopropyl-3,4-dihydroisoquinolin-7-yl)cycl...)
Affinity DataKi:  53nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Sus scrofa)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157087(6-(2-Phenyl-cyclopropyl)-8-(pyrimidin-2-ylamino)-n...)
Affinity DataKi:  54nMAssay Description:Binding affinity value against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50157087(6-(2-Phenyl-cyclopropyl)-8-(pyrimidin-2-ylamino)-n...)
Affinity DataKi:  54nMAssay Description:Binding affinity value against kallikreinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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