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Found 22 with Last Name = 'nikolsky' and Initial = 'ee'
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50313079(3-Dimethylcarbamoyloxy-1-methyl-pyridinium; bromid...)
Affinity DataIC50:  350nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189893(CHEMBL3828679)
Affinity DataIC50:  460nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189893(CHEMBL3828679)
Affinity DataIC50:  590nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50313079(3-Dimethylcarbamoyloxy-1-methyl-pyridinium; bromid...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189894(CHEMBL3827011)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189894(CHEMBL3827011)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189895(CHEMBL3828028)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189895(CHEMBL3828028)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189896(CHEMBL3827624)
Affinity DataIC50:  1.10E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189892(CHEMBL3827856)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189888(CHEMBL3827449)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189891(CHEMBL3828644)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189887(CHEMBL3827347)
Affinity DataIC50:  2.60E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189889(CHEMBL3828273)
Affinity DataIC50:  2.80E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189896(CHEMBL3827624)
Affinity DataIC50:  3.10E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189892(CHEMBL3827856)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189888(CHEMBL3827449)
Affinity DataIC50:  4.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189890(CHEMBL3828739)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of human AChE assessed as acetylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2 mins by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189889(CHEMBL3828273)
Affinity DataIC50:  8.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189887(CHEMBL3827347)
Affinity DataIC50:  9.00E+5nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189891(CHEMBL3828644)
Affinity DataIC50:  1.03E+6nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholinesterase(Homo sapiens (Human))
Kazan (Volga Region) Federal University

Curated by ChEMBL
LigandPNGBDBM50189890(CHEMBL3828739)
Affinity DataIC50:  1.19E+6nMAssay Description:Inhibition of human plasma BChE assessed as butyrylthiocholine hydrolysis preincubated for 10 mins followed by addition of substrate measured after 2...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed